Report error Found 3 Enz. Inhib. hit(s) for PDB: 8B8X
TargetPeroxisome proliferator-activated receptor gamma(Human)
The Scripps Research Institute
US Patent
The Scripps Research Institute
US Patent
Affinity DataIC50: 0.200nMAssay Description:The assay was performed according to manufacturer protocol. A mixture of 5 nM GST-PPARG-LBD, 5 nM Tb-GST-antibody, 5 nM Fluormone Pan- PPAR Green, an...More data for this Ligand-Target Pair
3D Structure (crystal)TargetPeroxisome proliferator-activated receptor gamma(Human)
The Scripps Research Institute
US Patent
The Scripps Research Institute
US Patent
Affinity DataIC50: 12nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
The Scripps Research Institute
US Patent
The Scripps Research Institute
US Patent
Affinity DataIC50: 263nMAssay Description:The assay was performed according to manufacturer protocol. A mixture of 5 nM GST-PPARG-LBD, 5 nM Tb-GST-antibody, 5 nM Fluormone Pan- PPAR Green, an...More data for this Ligand-Target Pair