Report error Found 2 Enz. Inhib. hit(s) for PDB: 8DKN
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Mit and Harvard
Curated by ChEMBL
Institute of Mit and Harvard
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair
3D Structure (crystal)TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Mit and Harvard
Curated by ChEMBL
Institute of Mit and Harvard
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair