Report error Found 1 Enz. Inhib. hit(s) for PDB: 8J1H
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Asahi Kasei Medical
Curated by ChEMBL
Asahi Kasei Medical
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair

3D Structure (crystal)