Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 8JLZ
Target5-hydroxytryptamine receptor 6(Rat)
University of Caen Normandie

Curated by ChEMBL
LigandPNGBDBM50171234([2-(5-Chloro-2-methyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H] lysergic acid diethylamide from rat 5-HT6 receptor transfected in HEK293 cells after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 6(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171234([2-(5-Chloro-2-methyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]LSD binding to cloned human 5-hydroxytryptamine 6 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 6(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171234([2-(5-Chloro-2-methyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)