Report error Found 4 Enz. Inhib. hit(s) for PDB: 8PJ8
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
Max Planck Institute of Psychiatry
Curated by ChEMBL
Max Planck Institute of Psychiatry
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
Max Planck Institute of Psychiatry
Curated by ChEMBL
Max Planck Institute of Psychiatry
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of iFit-FL from FKBP51 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
Max Planck Institute of Psychiatry
Curated by ChEMBL
Max Planck Institute of Psychiatry
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity to FKBP51 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
Max Planck Institute of Psychiatry
Curated by ChEMBL
Max Planck Institute of Psychiatry
Curated by ChEMBL
Affinity DataKd: 9.80nMAssay Description:Binding affinity to FKBP51 FK1 domain (unknown origin) assessed as dissociation constant at 25 degreeC by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair

3D Structure (crystal)