Report error Found 2 Enz. Inhib. hit(s) for PDB: 8T1D
TargetTransient receptor potential cation channel subfamily V member 4(Mouse)
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Mouse)
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Agonist activity at mouse TRPV4More data for this Ligand-Target Pair

3D Structure (crystal)