Compile Data Set for Download or QSAR
Report error Found 799 of affinity data for UniProtKB/TrEMBL: P00489
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50133435(4-(2-Chloro-phenyl)-1-ethyl-6-methyl-1,4-dihydro-p...)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50497973(CHEMBL3323454)
Affinity DataIC50: 7nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase a assessed as inhibition of release of phosphate from glucose-1-phosphate after 30 mins by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50382964(CHEMBL2030481)
Affinity DataIC50: 24nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50148913(CHEMBL3770455)
Affinity DataKi:  31nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-b using alpha-D-glucose-1-phosphate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50497969(CHEMBL3323453)
Affinity DataIC50: 45nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase a assessed as inhibition of release of phosphate from glucose-1-phosphate after 30 mins by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50148913(CHEMBL3770455)
Affinity DataKi:  65nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-a assessed as release of inorganic phosphate using varying levels of glucose-1-phospha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50241632(CHEMBL4101331)
Affinity DataKi:  125nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-a in presence of varying levels of glucose-1-phosphate and constant concentration of g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2019
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263826((1S)-1,5-Anhydro-D-glucitol-spiro[1.5]-3-(2-naphth...)
Affinity DataKi:  160nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263826((1S)-1,5-Anhydro-D-glucitol-spiro[1.5]-3-(2-naphth...)
Affinity DataKi:  160nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50196903(CHEMBL3916767)
Affinity DataIC50: 178nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using 10 mM of glucose-1-phosphate as substrate preincubated for 60 mins followed by substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50241632(CHEMBL4101331)
Affinity DataKi:  191nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-b in presence of varying levels of glucose-1-phosphate and constant concentration of g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2019
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50334099(2-((4R,5R,8R,9R,10R,13S,14R,15R)-4-(carboxymethyl)...)
Affinity DataIC50: 210nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50148915(CHEMBL3770514)
Affinity DataKi:  226nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-a assessed as release of inorganic phosphate using varying levels of glucose-1-phospha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50148915(CHEMBL3770514)
Affinity DataKi:  280nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-b using alpha-D-glucose-1-phosphate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataIC50: 330nMAssay Description:Inhibition of phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataKi:  342nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylase in presence of glycogen and 45 mM phosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263773(1-(2-naphthoyl)-3-((2R,3R,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataKi:  350nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263773(1-(2-naphthoyl)-3-((2R,3R,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataKi:  350nMpH: 6.8Assay Description:Inhibition of rabbit muscle glycogen phosphorylase b assessed as inorganic phosphate release at pH 6.8More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263773(1-(2-naphthoyl)-3-((2R,3R,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataKi:  350nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263773(1-(2-naphthoyl)-3-((2R,3R,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataKi:  350nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50263773(1-(2-naphthoyl)-3-((2R,3R,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataKi:  350nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataIC50: 390nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataKi:  396nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylase in presence of 6.17 mM glycogen and phosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50016703(CHEMBL80254 | Imino-D-Arabinitol | BDBM50031485 | ...)
Affinity DataKi:  400nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase using tritium-labeled glycogen as substrate by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50437354(CHEMBL2408225)
Affinity DataKi:  410nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50437354(CHEMBL2408225)
Affinity DataKi:  410nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50430005(FR258900 | CHEMBL1234956)
Affinity DataKi:  460nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM34110(glucopyranosylidene-spiro-isoxazoline, 4e)
Affinity DataKi:  630nM ΔG°:  -36.0kJ/molepH: 6.8 T: 2°CAssay Description:Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM34110(glucopyranosylidene-spiro-isoxazoline, 4e)
Affinity DataIC50: 630nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50009082(CHEMBL3237972)
Affinity DataKi:  670nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50056223(CHEMBL3322301)
Affinity DataKi:  700nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50182801(CHEMBL206468 | AFEGOSTAT TARTRATE | D-Isofagomine ...)
Affinity DataIC50: 760nMAssay Description:Inhibition of phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50312225(CHEMBL4161353)
Affinity DataKi:  780nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50312361(CHEMBL4169281)
Affinity DataKi:  840nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50194702((3R,4R,5R)-5-(HYDROXYMETHYL)-1-(3-PHENYLPROPYL)PIP...)
Affinity DataIC50: 840nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50382963(CHEMBL2030480)
Affinity DataIC50: 900nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50313014(CHEMBL4172670)
Affinity DataKi:  980nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50386288(CHEMBL2041081)
Affinity DataKi:  1.02E+3nMAssay Description:Competitive inhibition of rabbit skeletal muscle glycogen phosphorylase b using Glc-1-P as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50346702(CHEMBL574993)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50346702(CHEMBL574993)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase a assessed as glycogen synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50346677(CHEMBL1796866)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50312361(CHEMBL4169281)
Affinity DataKi:  1.19E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-b assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50310522(2alpha-Hydroxyurs-12-en-28-oic acid | CHEMBL107884...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase assessed as release of phosphate from glucose-1-phosphate after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50182801(CHEMBL206468 | AFEGOSTAT TARTRATE | D-Isofagomine ...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50346595(CHEMBL1797018)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50346692(CHEMBL1797010)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50146082(CHEMBL3763876)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50009074(CHEMBL3237966)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50056224(CHEMBL3322302)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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