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Report error Found 99 for UniProtKB: P03428
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615249(CHEMBL5289925)
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050703(CHEMBL3318000)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050702(CHEMBL3317999)
Affinity DataKd:  30nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050701(CHEMBL3317986)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050700(CHEMBL3317985)
Affinity DataKd:  200nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050699(CHEMBL3317984)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050698(CHEMBL3317983)
Affinity DataKd:  200nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050697(CHEMBL3317982)
Affinity DataKd:  70nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50633335(CHEMBL5419341)
Affinity DataKd:  202nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50633334(CHEMBL5433576)
Affinity DataKd:  145nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50633332(CHEMBL5397789)
Affinity DataKd:  46nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50633331(CHEMBL5429336)
Affinity DataKd:  468nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050705(CHEMBL3318001)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615248(CHEMBL5280401)
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615247(CHEMBL5283800)
Affinity DataKd:  3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615246(CHEMBL5280871)
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615245(CHEMBL5279168)
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615244(CHEMBL5289034)
Affinity DataKd:  150nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615243(CHEMBL5281405)
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50615242(CHEMBL5272653)
Affinity DataKd:  200nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50586991(CHEMBL5094914)
Affinity DataKd:  1.60E+3nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50586989(CHEMBL5075807)
Affinity DataKd:  6.40E+3nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50586988(CHEMBL5087029)
Affinity DataKd:  580nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050718(CHEMBL3317969)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050760(CHEMBL3317981)
Affinity DataKd:  70nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050759(CHEMBL3317980)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050758(CHEMBL3317979)
Affinity DataKd:  4.90E+3nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050757(CHEMBL3317978)
Affinity DataKd:  90nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050756(CHEMBL3317977)
Affinity DataKd:  80nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050754(CHEMBL3317976)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050750(CHEMBL3317975)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050722(CHEMBL3317974)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050721(CHEMBL3317973)
Affinity DataKd:  300nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050720(CHEMBL3317972)
Affinity DataKd:  700nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050719(CHEMBL3317970)
Affinity DataKd:  300nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50586990(CHEMBL5091340)
Affinity DataKd:  110nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050717(CHEMBL3317991)
Affinity DataKd:  90nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050716(CHEMBL3317990)
Affinity DataKd:  20nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050715(CHEMBL3317989)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050714(CHEMBL3317988)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050713(CHEMBL3317987)
Affinity DataKd:  500nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050710(CHEMBL3318006)
Affinity DataKd: <5nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050709(CHEMBL3318005)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050708(CHEMBL3318004)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050707(CHEMBL3318003)
Affinity DataKd:  9nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050706(CHEMBL3318002)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50507228(CHEMBL4434862)
Affinity DataEC50:  0.5nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM62536(cid_646771 | 2-[(2-phenyl-[1]benzofuro[3,2-d]pyrim...)
Affinity DataKd:  250nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50507238(CHEMBL4527175)
Affinity DataEC50:  12nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50507237(CHEMBL4567152)
Affinity DataEC50:  13nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
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