Compile Data Set for Download or QSAR
Report error Found 135 of affinity data for UniProtKB/TrEMBL: P15101
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(CHEMBL433493 | 1-(3,5-Difluoro-4-hydroxy-benzyl)-1...)
Affinity DataKi:  5.70nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014970(CHEMBL351873 | 4-(3,5-Difluoro-4-hydroxy-benzyl)-2...)
Affinity DataIC50: 35nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50548688(CHEMBL4764135)
Affinity DataIC50: 39nMAssay Description:Inhibition of bovine adrenal medulla DBH incubated for 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014983(CHEMBL278068 | 1-(3,5-Difluoro-benzyl)-1,3-dihydro...)
Affinity DataKi:  41nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(CHEMBL24510 | 5-Butyl-pyridine-2-carboxylic acid |...)
Affinity DataIC50: 50nMAssay Description:Inhibition of bovine adrenal medulla DBH incubated for 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(CHEMBL164747 | 4-(2-Mercapto-imidazol-1-ylmethyl)-...)
Affinity DataKi:  55nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(CHEMBL164747 | 4-(2-Mercapto-imidazol-1-ylmethyl)-...)
Affinity DataKi:  55nMpH: 4.5Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(CHEMBL433493 | 1-(3,5-Difluoro-4-hydroxy-benzyl)-1...)
Affinity DataIC50: 74nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(CHEMBL433493 | 1-(3,5-Difluoro-4-hydroxy-benzyl)-1...)
Affinity DataIC50: 74nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (0.060-0.0877).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015622(CHEMBL275322 | 1-(2-Thiophen-2-yl-ethyl)-1,3-dihyd...)
Affinity DataIC50: 114nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015620(CHEMBL54434 | 1-(2-Thiophen-3-yl-ethyl)-1,3-dihydr...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(CHEMBL24510 | 5-Butyl-pyridine-2-carboxylic acid |...)
Affinity DataKi:  149nMAssay Description:Inhibition of Dopamine beta hydroxylase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(CHEMBL24510 | 5-Butyl-pyridine-2-carboxylic acid |...)
Affinity DataKi:  149nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014983(CHEMBL278068 | 1-(3,5-Difluoro-benzyl)-1,3-dihydro...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(CHEMBL164747 | 4-(2-Mercapto-imidazol-1-ylmethyl)-...)
Affinity DataKi:  344nMpH: 6.6Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 6.6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015617(CHEMBL54906 | 1-[2-(5-Methyl-thiophen-2-yl)-ethyl]...)
Affinity DataIC50: 491nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014963(CHEMBL165242 | 1-(3,5-Difluoro-4-hydroxy-benzyl)-1...)
Affinity DataIC50: 660nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025811(1-(3,5-Dichloro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50: 680nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (25-81).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015621(CHEMBL55949 | 1-(5-Chloro-thiophen-2-ylmethyl)-1,3...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014984(CHEMBL165150 | 4-(3,5-Difluoro-benzyl)-2,4-dihydro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014983(CHEMBL278068 | 1-(3,5-Difluoro-benzyl)-1,3-dihydro...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (1.0-1.9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014983(CHEMBL278068 | 1-(3,5-Difluoro-benzyl)-1,3-dihydro...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014971(CHEMBL352449 | 1-(3,5-Difluoro-benzyl)-imidazolidi...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025795(1-(3-Fluoro-4-hydroxy-benzyl)-1,3-dihydro-imidazol...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (0.9-2.2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014967(CHEMBL165032 | 1-(3,5-Difluoro-benzyl)-1H-tetrazol...)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015619(CHEMBL54500 | 1-(3-Thiophen-2-yl-propyl)-1,3-dihyd...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014979(CHEMBL165206 | 4-(3-Fluoro-benzyl)-2,4-dihydro-[1,...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025806(1-(3-Chloro-4-hydroxy-benzyl)-1,3-dihydro-imidazol...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (1.7-2.4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025798(1-[3-(3,5-Dichloro-phenyl)-propyl]-1,3-dihydro-imi...)
Affinity DataIC50: 2.10E+3nMAssay Description:Percent inhibition against bovine Dopamine beta hydroxylase at 10E-4 M concentration of the compound; Range is between (1.8-2.6).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014962(CHEMBL350128 | 1-[3-(4-Hydroxy-phenyl)-propyl]-1,3...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Dopamine beta hydroxylase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014962(CHEMBL350128 | 1-[3-(4-Hydroxy-phenyl)-propyl]-1,3...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025803(1-(3,4-Dihydroxy-benzyl)-1,3-dihydro-imidazole-2-t...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (1.1-3.8).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025793(1-(3,5-Dichloro-benzyl)-1,3-dihydro-imidazole-2-th...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (1.9-3.0)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(CHEMBL164747 | 4-(2-Mercapto-imidazol-1-ylmethyl)-...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (1.3-4.6)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(CHEMBL164747 | 4-(2-Mercapto-imidazol-1-ylmethyl)-...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(CHEMBL164747 | 4-(2-Mercapto-imidazol-1-ylmethyl)-...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Dopamine beta hydroxylase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014976(CHEMBL351468 | 1-(3,5-Difluoro-benzyl)-1H-pyrimidi...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015624(CHEMBL442739 | 1-(4-Thiophen-2-yl-butyl)-1,3-dihyd...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014982(CHEMBL351936 | 1-(3-Fluoro-benzyl)-imidazolidine-2...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015627(CHEMBL417921 | 1-(5-Fluoro-thiophen-2-ylmethyl)-1,...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50025792(1-[3-(3,5-Difluoro-phenyl)-propyl]-1,3-dihydro-imi...)
Affinity DataIC50: 4.70E+3nMAssay Description:Percent inhibition against bovine Dopamine beta hydroxylase at 10E-4 M concentration of the compound; Range is between (4.2-5.3).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015626(CHEMBL294141 | 1-Thiophen-2-ylmethyl-1,3-dihydro-i...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50017831(CHEMBL163500 | 2-[1,3]Dithiolan-2-ylidene-ethylami...)
Affinity DataKi:  5.00E+3nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015625(CHEMBL55206 | 1-Thiophen-3-ylmethyl-1,3-dihydro-im...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014969(CHEMBL63907 | 1-(3-Fluoro-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (4.9-6.5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014969(CHEMBL63907 | 1-(3-Fluoro-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015623(CHEMBL55205 | 1-(5-Methyl-thiophen-2-ylmethyl)-1,3...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014959(CHEMBL350557 | 1-(3,5-Difluoro-benzyl)-1,3-dihydro...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50014973(CHEMBL165154 | 2-(3,5-Difluoro-benzyl)-2,4-dihydro...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDopamine beta-hydroxylase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50015618(CHEMBL55767 | 1-Furan-2-ylmethyl-1,3-dihydro-imida...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibitory activity against bovine adrenal dopamine beta-hydroxylase (DBH)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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