Compile Data Set for Download or QSAR
Report error Found 27 for UniProtKB: P97717
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50060964BDBM50060964(5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 39687BDBM39687(cid_5717105 | MLS000532635 | SMR000137574 | CHEMBL...)
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280816BDBM50280816(N-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280824BDBM50280824(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280829BDBM50280829(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280831BDBM50280831(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280815BDBM50280815(N-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280826BDBM50280826(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280830BDBM50280830(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280822BDBM50280822(4-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280825BDBM50280825(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280817BDBM50280817(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280818BDBM50280818(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280827BDBM50280827(1'-{2-[4-(5-fluoro-1H-3-indolylmethyl)hexahydro-1-...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280823BDBM50280823(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280820BDBM50280820(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280828BDBM50280828(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280819BDBM50280819(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280821BDBM50280821(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280832BDBM50280832(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270777BDBM50270777(CHEMBL4126353)
Affinity DataIC50: 348nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270778BDBM50270778(CHEMBL4126498)
Affinity DataIC50: 577nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270779BDBM50270779(CHEMBL4129778)
Affinity DataIC50: 711nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078561BDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270772BDBM50270772(CHEMBL4128701)
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dundee

US Patent
LigandChemical structure of BindingDB Monomer ID 186935BDBM186935(US9079895, 23s)
Affinity DataKi:  6.64E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

TargetAlpha-1B adrenergic receptor(Mouse)
University of Dundee

US Patent
LigandChemical structure of BindingDB Monomer ID 186927BDBM186927(US9079895, 19s)
Affinity DataKi:  7.21E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent