Compile Data Set for Download or QSAR
Report error Found 214 of affinity data for UniProtKB/TrEMBL: Q6P5T3
LigandChemical structure of BindingDB Monomer ID 50391858BDBM50391858(CHEMBL2147281)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391863BDBM50391863(CHEMBL2147286)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391867BDBM50391867(CHEMBL2147290)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391860BDBM50391860(CHEMBL2147283)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204367BDBM50204367(dirlotapide | CHEMBL410414)
Affinity DataIC50: 0.0110nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098322BDBM50098322(9-(4-{5-Methyl-4-[(4'-trifluoromethyl-biphenyl-2-c...)
Affinity DataIC50: 0.0200nMAssay Description:In vitro inhibition of human microsomal triglyceride transfer protein in HepG2 cells using apoB secretion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391875BDBM50391875(CHEMBL2147296)
Affinity DataIC50: 0.0210nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391876BDBM50391876(CHEMBL2147292)
Affinity DataIC50: 0.0250nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098321BDBM50098321(9-(4-{2,5-Dimethyl-4-[(4'-trifluoromethyl-biphenyl...)
Affinity DataIC50: 0.0300nMAssay Description:In vitro inhibition of human microsomal triglyceride transfer protein in HepG2 cells using apoB secretion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391866BDBM50391866(CHEMBL2147294)
Affinity DataIC50: 0.0580nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098326BDBM50098326(9-(4-{2-Isopropyl-4-[(4'-trifluoromethyl-biphenyl-...)
Affinity DataIC50: 0.0600nMAssay Description:In vitro inhibition of human microsomal triglyceride transfer protein in HepG2 cells using apoB secretion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391877BDBM50391877(CHEMBL2147293)
Affinity DataIC50: 0.0660nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391869BDBM50391869(CHEMBL2147301)
Affinity DataIC50: 0.101nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391871BDBM50391871(CHEMBL2147298)
Affinity DataIC50: 0.105nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391872BDBM50391872(CHEMBL2147299)
Affinity DataIC50: 0.122nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098324BDBM50098324(9-(4-{2-Methyl-4-[(4'-trifluoromethyl-biphenyl-2-c...)
Affinity DataIC50: 0.150nMAssay Description:In vitro inhibition of human microsomal triglyceride transfer protein in HepG2 cells using apoB secretion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098325BDBM50098325(9-(4-{4-[(4'-Trifluoromethyl-biphenyl-2-carbonyl)-...)
Affinity DataIC50: 0.240nMAssay Description:In vitro inhibition of human microsomal triglyceride transfer protein in HepG2 cells using apoB secretion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391874BDBM50391874(CHEMBL2147295)
Affinity DataIC50: 0.253nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391857BDBM50391857(CHEMBL2147280)
Affinity DataIC50: 0.345nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391856BDBM50391856(CHEMBL2147279)
Affinity DataIC50: 0.378nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391862BDBM50391862(CHEMBL2147285)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391870BDBM50391870(CHEMBL2147300)
Affinity DataIC50: 0.484nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as unbound drug level causing inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391861BDBM50391861(CHEMBL2147284)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391875BDBM50391875(CHEMBL2147296)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277189BDBM50277189((R)-6-methyl-N-(2-(thiazol-2-ylmethylamino)-2,3-di...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as apolipoprotein B production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391863BDBM50391863(CHEMBL2147286)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391869BDBM50391869(CHEMBL2147301)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391858BDBM50391858(CHEMBL2147281)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391867BDBM50391867(CHEMBL2147290)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098320BDBM50098320(9-(4-{4-[(4'-Trifluoromethyl-biphenyl-2-carbonyl)-...)
Affinity DataIC50: 0.800nMAssay Description:In vitro inhibition of human microsomal triglyceride transfer protein in HepG2 cells using apoB secretion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391865BDBM50391865(CHEMBL2147291)
Affinity DataIC50: 0.830nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50107789BDBM50107789((R)-methyl 5-(6-methyl-4'-(trifluoromethyl)bipheny...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as apolipoprotein B production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098321BDBM50098321(9-(4-{2,5-Dimethyl-4-[(4'-trifluoromethyl-biphenyl...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of human Microsomal Triglyceride Transfer Protein, (triglyceride transfer assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098322BDBM50098322(9-(4-{5-Methyl-4-[(4'-trifluoromethyl-biphenyl-2-c...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of human Microsomal Triglyceride Transfer Protein, (triglyceride transfer assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098324BDBM50098324(9-(4-{2-Methyl-4-[(4'-trifluoromethyl-biphenyl-2-c...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of human Microsomal Triglyceride Transfer Protein, (triglyceride transfer assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184105BDBM50184105(4'-trifluoromethyl-biphenyl-2-carboxylic acid (4-{...)
Affinity DataIC50: 1.01nMAssay Description:Inhibition of MTP in canine liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391876BDBM50391876(CHEMBL2147292)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391873BDBM50391873(CHEMBL2147297)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391873BDBM50391873(CHEMBL2147297)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391868BDBM50391868(CHEMBL2146489)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391864BDBM50391864(CHEMBL2147287)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391868BDBM50391868(CHEMBL2146489)
Affinity DataIC50: 1.21nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391857BDBM50391857(CHEMBL2147280)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184109BDBM50184109(4'-trifluoromethyl-biphenyl-2-carboxylic acid {2-m...)
Affinity DataIC50: 1.64nMAssay Description:Inhibition of MTP in canine liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184153BDBM50184153(4'-trifluoromethyl-biphenyl-2-carboxylic acid (4-{...)
Affinity DataIC50: 1.68nMAssay Description:Inhibition of MTP in canine liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184111BDBM50184111(4'-trifluoromethyl-biphenyl-2-carboxylic acid [2-m...)
Affinity DataIC50: 1.75nMAssay Description:Inhibition of MTP in canine liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184165BDBM50184165(4'-trifluoromethyl-biphenyl-2-carboxylic acid (4-{...)
Affinity DataIC50: 1.78nMAssay Description:Inhibition of MTP in canine liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50391856BDBM50391856(CHEMBL2147279)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of MTP in human HepG2 cells assessed as inhibition of apoB secretion after 40 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184118BDBM50184118(4'-trifluoromethyl-biphenyl-2-carboxylic acid {2-m...)
Affinity DataIC50: 2nMAssay Description:Inhibition of MTP in canine liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50098323BDBM50098323(9-(4-{2-Propyl-4-[(4'-trifluoromethyl-biphenyl-2-c...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of human Microsomal Triglyceride Transfer Protein, (triglyceride transfer assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 214 total ) | Next | Last >>
Jump to: