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Found 8 of affinity data for UniProtKB/TrEMBL: D3Z7P3
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM109086(US10793535, Cmpd ID 727 | US8604016, 670 | US99382...)
Affinity DataIC50:  20nMAssay Description:Inhibition of GLS1 in mouse kidney assessed as inhibition of glutamate production using glutamine as substrate incubated for 1 hr by coupled assayMore data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM109086(US10793535, Cmpd ID 727 | US8604016, 670 | US99382...)
Affinity DataIC50:  20nMAssay Description:Inhibition of GLS1 in mouse brain assessed as inhibition of glutamate production using glutamine as substrate incubated for 1 hr by coupled assayMore data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503321(CHEMBL4540444)
Affinity DataIC50: <25nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503294(CHEMBL4577734)
Affinity DataIC50: <50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503291(CHEMBL4562029)
Affinity DataIC50:  50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation using glutamine as substrate by Nessler's reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503289(CHEMBL4462220)
Affinity DataIC50:  50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503296(CHEMBL4452754)
Affinity DataIC50: <50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503312(CHEMBL4537860)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed