TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 18nMAssay Description:Binding constant for PIP5K1C kinase domainMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of N-terminal His6-tagged full length recombinant human PIP5K1gamma by microfluidic mobility shift assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 77nMAssay Description:Binding affinity to PIP5K1C (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 130nMAssay Description:Binding constant for PIP5K1C kinase domainMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of PIP5Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal 6His-tagged full-length recombinant human PIP5K1C expressed in baculovirus infected Sf21 cells using PI4P/PS as substrate in...More data for this Ligand-Target Pair

















































