TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 350nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 430nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 510nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 1.19E+4nMAssay Description:Binding affinity to biotinylated STK16 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity to C-terminal AVI-tagged STK16 (unknown origin) (13 to 305 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 5.10E+4nMAssay Description:Binding affinity to C-terminal AVI-tagged STK16 (unknown origin) (13 to 305 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to C-terminal AVI-tagged STK16 (unknown origin) (13 to 305 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of human STK16 in presence of [gamma-33P-ATP] by radiometric scintillation assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of human STK16 in presence of [gamma-33P-ATP] by radiometric scintillation assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of MPSK1 (unknown origin) by biochemical assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of human wild type partial length STK16 (G11 to I305) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 235nMAssay Description:Inhibition of human STK16 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 242nMAssay Description:Inhibition of human STK16 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 295nMAssay Description:The enzymatic assay was performed using the LifeTechnology SelectScreen.More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 885nMAssay Description:Inhibition of STK16 (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of MPSK1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of recombinant full length His-tagged human STK16 expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory concentration against cyclin dependent kinase-2 (CDK2)/Cyclin EMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human STK16 in presence of 10 uM ATP by radiometric analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair