Compile Data Set for Download or QSAR
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Found 4 of affinity data for UniProtKB/TrEMBL: P05183
TargetCytochrome P450 3A2(RAT)
Pudue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A2(RAT)
Pudue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)
Affinity DataKi:  1.42E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetCytochrome P450 3A2(RAT)
Pudue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  5.26E+4nMAssay Description:Inhibition of CYP3A2 in rat liver microsomes using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A2(RAT)
Pudue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)
Affinity DataIC50:  2.32E+4nMMore data for this Ligand-Target Pair
In DepthDetails