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Found 170 for UniProtKB: P08263
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50054198(CHEMBL3310888)
Affinity DataKi:  360nMAssay Description:Competitive inhibition of human GSTA1 activity by double reciprocal Lineweaver-Burk graphMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50054196(CHEMBL3310887)
Affinity DataKi:  380nMAssay Description:Competitive inhibition of human GSTA1 activity by double reciprocal Lineweaver-Burk graphMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043758(2-Amino-4-[1-(carboxymethyl-carbamoyl)-2-hexylsulf...)
Affinity DataKi:  840nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50054194(CHEMBL3310886)
Affinity DataKi:  1.47E+3nMAssay Description:Competitive inhibition of human GSTA1 activity by double reciprocal Lineweaver-Burk graphMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50295556(C6H5-SO2-Glu-Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-G...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by 1-chloro-2,4-dinitrobenzene competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50295554(C6H5-SO2-Glu-Gln-Ser-Leu-Gly-Asn-Gln-Trp-Ala-Arg-G...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by 1-chloro-2,4-dinitrobenzene competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50295555(C6H5-SO2-Glu-Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-G...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by 1-chloro-2,4-dinitrobenzene competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50054205(CHEMBL3310889)
Affinity DataKi:  1.75E+3nMAssay Description:Competitive inhibition of human GSTA1 activity by double reciprocal Lineweaver-Burk graphMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043764(2-Amino-4-{1-[(carboxy-phenyl-methyl)-carbamoyl]-2...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50295556(C6H5-SO2-Glu-Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-G...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by glutathione competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50295554(C6H5-SO2-Glu-Gln-Ser-Leu-Gly-Asn-Gln-Trp-Ala-Arg-G...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by glutathione competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50295555(C6H5-SO2-Glu-Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-G...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by glutathione competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043760(2-Amino-4-[1-[(carboxy-phenyl-methyl)-carbamoyl]-2...)
Affinity DataKi:  1.47E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043762(2-Amino-4-{2-benzylsulfanyl-1-[(carboxy-phenyl-met...)
Affinity DataKi:  2.43E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043761(2-Amino-4-[1-(2-carboxy-ethylcarbamoyl)-2-hexylsul...)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043763(2-Amino-4-[1-(2-carboxy-ethylcarbamoyl)-2-(4-methy...)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50395590(CHEMBL2165141)
Affinity DataKi:  7.10E+4nMAssay Description:Competitive inhibition of recombinant human GSTA1-1 expressed in Escherichia coli BL21 (DE3) using CDNB as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50395591(CHEMBL2165146)
Affinity DataKi:  1.35E+5nMAssay Description:Competitive inhibition of recombinant human GSTA1-1 expressed in Escherichia coli BL21 (DE3) using CDNB as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50043759(2-Amino-4-[2-benzylsulfanyl-1-(2-carboxy-ethylcarb...)
Affinity DataKi:  3.60E+5nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM218770(US9296757, 92)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218771(US9296757, 93)
Affinity DataIC50:  0.700nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218768(US9296757, 90)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218766(US9296757, 88)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218767(US9296757, 89)
Affinity DataIC50:  1.90nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218765(US9296757, 87)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218764(US9296757, 86)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218763(US9296757, 85)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218709(US9296757, 31)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214639(US9284319, 7)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214635(US9284319, 3)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214633(US9284319, 1)
Affinity DataIC50:  7nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218714(US9296757, 36)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218687(US9296757, 9)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214649(US9284319, R7 | US9730929, Example R7 | US9783543,...)
Affinity DataIC50:  11nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218688(US9296757, 10)
Affinity DataIC50:  11nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214638(US9284319, 6)
Affinity DataIC50:  12nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214649(US9284319, R7 | US9730929, Example R7 | US9783543,...)
Affinity DataIC50:  13nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214637(US9284319, 5)
Affinity DataIC50:  13nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50186225(3-((3-(2-(2,3-dichloro-4-(2-methylenebutanoyl)phen...)
Affinity DataIC50:  13.7nMAssay Description:Inhibition of GST A1-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM214639(US9284319, 7)
Affinity DataIC50:  14nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50186230(3-((4-(2-(2,3-dichloro-4-(2-methylenebutanoyl)phen...)
Affinity DataIC50:  14.3nMAssay Description:Inhibition of GST A1-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM214640(US9284319, 8)
Affinity DataIC50:  15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214636(US9284319, 4)
Affinity DataIC50:  15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214641(US9284319, 9)
Affinity DataIC50:  15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218708(US9296757, 30 | US9296757, 33)
Affinity DataIC50:  15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214635(US9284319, 3)
Affinity DataIC50:  17nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214648(US9284319, R6 | US9730929, Example R6 | US9783543,...)
Affinity DataIC50:  17nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214640(US9284319, 8)
Affinity DataIC50:  19nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM218747(US9296757, 69)
Affinity DataIC50:  19nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM214633(US9284319, 1)
Affinity DataIC50:  19nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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