Compile Data Set for Download or QSAR
maximum 50k data
Found 28 of affinity data for UniProtKB/TrEMBL: P0A8L1
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339906(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Seryl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichia...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458116(CHEMBL4208640)
Affinity DataKi:  523nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Seryl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichia...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339906(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataIC50:  210nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339906(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataIC50:  210nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530866(CHEMBL4529844)
Affinity DataIC50:  450nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530866(CHEMBL4529844)
Affinity DataIC50:  450nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530864(CHEMBL4467050)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530864(CHEMBL4467050)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530862(CHEMBL4446951)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530862(CHEMBL4446951)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataIC50:  6.65E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataIC50:  6.65E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530861(CHEMBL4452350)
Affinity DataIC50:  9.38E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530861(CHEMBL4452350)
Affinity DataIC50:  9.38E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530860(CHEMBL4461782)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530860(CHEMBL4461782)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530863(CHEMBL4449289)
Affinity DataIC50:  3.62E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530863(CHEMBL4449289)
Affinity DataIC50:  3.62E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530865(CHEMBL4471342)
Affinity DataIC50:  2.85E+5nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530865(CHEMBL4471342)
Affinity DataIC50:  2.85E+5nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339906(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as dissociation constant by isoth...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataKd:  1.92E+3nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as affinity constant for second b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataKd:  290nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as dissociation constant by isoth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataKd:  290nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as affinity constant for first bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataKd:  290nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as dissociation constant by isoth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339906(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as dissociation constant by isoth...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataKd:  1.92E+3nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as affinity constant for second b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50530859(CHEMBL4561900)
Affinity DataKd:  290nMAssay Description:Binding affinity to C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) SerRS assessed as affinity constant for first bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB