TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.182nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.204nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparationMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.347nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.692nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Displacement of [3H]-RX821002 from adrenergic alpha 2 receptor in human brain membrane by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.912nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.912nMAssay Description:Displacement of [3H]RX821002 from adrenergic alpha2 receptor in human brain frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.912nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenoceptor in human prefrontal cortex neural membrane after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]RX 821002 from human recombinant adrenergic alpha-2B receptor expressed in CHO cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparationMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparationMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to alpha2 adrenoceptor in human cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]RX821002 from alpha-2 adrenergic receptor in human brain pre-frontal cortex neural membranes after 30 mins by liquid scintillatio...More data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-RX821002 from adrenergic alpha 2 receptor in human brain membrane by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]RX821002 from adrenergic alpha2 receptor in human brain frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-RX821002 from adrenergic alpha 2 receptor in human brain membrane by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.91nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro binding affinity towards human alpha-2B adrenergic receptor using [3H]-rauwolscineMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of HT-29 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparationMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.82nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair