Compile Data Set for Download or QSAR
Report error Found 9430 of affinity data for UniProtKB/TrEMBL: P22303
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093582(CHEMBL3585782)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093588(CHEMBL3585776)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093587(CHEMBL3585777)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50049862(CHEMBL3322232)
Affinity DataIC50: 0.00600nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093581(CHEMBL3585783)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093589(CHEMBL3585775)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093583(CHEMBL3585781)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50523376(CHEMBL4589980)
Affinity DataIC50: 0.00800nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093597(CHEMBL3585784)
Affinity DataKi:  0.00800nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM9012(7-[(6,8-dichloro-1,2,3,4-tetrahydroacridin-9-yl)am...)
Affinity DataIC50: 0.00800nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The absorbance changes at 412 nm were recorded for 5 min with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM9012(7-[(6,8-dichloro-1,2,3,4-tetrahydroacridin-9-yl)am...)
Affinity DataIC50: 0.00800nMAssay Description:Inhibition of human AchEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093585(CHEMBL3585779)
Affinity DataKi:  0.0110nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456700(CHEMBL4205425)
Affinity DataIC50: 0.0110nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50271367(N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[...)
Affinity DataKi:  0.0120nMAssay Description:Inhibition of human acetylcholine esteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50271367(N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[...)
Affinity DataKi:  0.0120nMAssay Description:Inhibition of human recombinant AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456689(CHEMBL4205954)
Affinity DataIC50: 0.0130nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456692(CHEMBL4209803)
Affinity DataIC50: 0.0140nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456691(CHEMBL4210316)
Affinity DataIC50: 0.0140nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456690(CHEMBL4217663)
Affinity DataIC50: 0.0140nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456693(CHEMBL4214430)
Affinity DataIC50: 0.0170nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456699(CHEMBL4213253)
Affinity DataIC50: 0.0190nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM9022(N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of human AchEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50318731(3-(1H-indol-3-yl)-N-(6-(1,2,3,4-tetrahydroacridin-...)
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456696(CHEMBL4214707)
Affinity DataIC50: 0.0210nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456682(CHEMBL4210041)
Affinity DataIC50: 0.0220nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093586(CHEMBL3585778)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM10597((1S)-7-chloro-15-ethyl-10-azatetracyclo[11.3.1.0^{...)
Affinity DataKi:  0.0260nM ΔG°:  -60.4kJ/molepH: 7.0 T: 2°CAssay Description:Assays were conducted at 25 C in 20 mM sodium phosphate buffer (pH 7.0) and 0.01% bovine serum albumin unless otherwise noted. AChE concentrations we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM10597((1S)-7-chloro-15-ethyl-10-azatetracyclo[11.3.1.0^{...)
Affinity DataKi:  0.0260nM ΔG°:  -60.4kJ/molepH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by E llman. Inhibition of enzyme activity was measured over a substrate c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456694(CHEMBL4205144)
Affinity DataIC50: 0.0260nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456688(CHEMBL4218191)
Affinity DataIC50: 0.0260nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50369748(CHEMBL208599)
Affinity DataKi:  0.0260nMAssay Description:Inhibitory activity against human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093583(CHEMBL3585781)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093582(CHEMBL3585782)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093585(CHEMBL3585779)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093584(CHEMBL3585780)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093588(CHEMBL3585776)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093586(CHEMBL3585778)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093587(CHEMBL3585777)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093581(CHEMBL3585783)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093589(CHEMBL3585775)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093597(CHEMBL3585784)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456687(CHEMBL4208866)
Affinity DataIC50: 0.0280nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50456698(CHEMBL4209518)
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50200340((+/-)-huprineY hydrochloride | (+/-)-huprine Y-HCl...)
Affinity DataKi:  0.0330nMAssay Description:Binding affinity to human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50380559(CHEMBL2019048)
Affinity DataIC50: 0.0350nMAssay Description:Inhibition of human erythrocytes AChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50093584(CHEMBL3585780)
Affinity DataKi:  0.0380nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as AChI hydrolysis using AChI and DTNB as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM9017(7-[(6,8-dichloro-1,2,3,4-tetrahydroacridin-9-yl)am...)
Affinity DataIC50: 0.0400nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The absorbance changes at 412 nm were recorded for 5 min with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50022775(m-Trimethylammoniumphenyldimethylcarbamate | Prost...)
Affinity DataIC50: 0.0430nMAssay Description:Inhibition of human acetylcholine esteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50634776(Donepezil | Donepezilo | D-797 | Donaz)
Affinity DataIC50: 0.0490nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetAcetylcholinesterase(Human)
Agriibrahim£E£En University

Curated by ChEMBL
LigandPNGBDBM50651582(CHEMBL5633243)
Affinity DataIC50: 0.0580nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
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