Compile Data Set for Download or QSAR
Report error Found 107 of affinity data for UniProtKB/TrEMBL: P29994
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323706(CHEMBL1212943)
Affinity DataKd:  0.140nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323704(CHEMBL1213158)
Affinity DataKd:  0.180nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323705(CHEMBL1213159)
Affinity DataKd:  0.180nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323709(CHEMBL1213163)
Affinity DataKd:  0.200nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323707(CHEMBL1213160)
Affinity DataKd:  0.200nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  0.210nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323710((1R,2R,3S,4R,6S)-3,6-dihydroxycyclohexane-1,2,4-tr...)
Affinity DataKd:  0.220nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323708(CHEMBL1213161)
Affinity DataKd:  0.330nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323707(CHEMBL1213160)
Affinity DataKd:  0.360nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323704(CHEMBL1213158)
Affinity DataKd:  0.410nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323706(CHEMBL1212943)
Affinity DataKd:  0.420nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323704(CHEMBL1213158)
Affinity DataKd:  0.450nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323705(CHEMBL1213159)
Affinity DataKd:  0.470nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323711((1R,2R,3S,4S,5R,6S)-5-(2-aminoethoxy)-3,6-dihydrox...)
Affinity DataKd:  0.520nMAssay Description:Displacement of [3H]IP3 from rat recombinant IP3R1 binding core residue (224-604) expressed in chicken DT40 cells by equilibrium competitive binding ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323705(CHEMBL1213159)
Affinity DataKd:  0.860nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323707(CHEMBL1213160)
Affinity DataKd:  0.890nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323706(CHEMBL1212943)
Affinity DataKd:  0.900nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataKd:  1.26nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50514586(CHEMBL4578747)
Affinity DataKd:  1.40nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataKd:  1.40nMAssay Description:Displacement of [3H]-IP3 from IP3R1 in Wistar rat cerebellar membrane measured after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50514586(CHEMBL4578747)
Affinity DataKd:  1.40nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323709(CHEMBL1213163)
Affinity DataKd:  1.63nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataEC50:  2.10nMAssay Description:Activity at rat IP3 type 1 receptor expressed in DT40 cell assessed as calcium ion mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50194703(5'-Deoxy-5'-phenyladenophostin A)
Affinity DataEC50:  2.10nMAssay Description:Activity at rat IP3 type 1 receptor expressed in DT40 cell assessed as calcium ion mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataEC50:  2.10nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  2.32nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50194704(5'-deoxy-5'-phenethyladenophostin A 2',3'',4''-tri...)
Affinity DataEC50:  2.70nMAssay Description:Activity at rat IP3 type 1 receptor expressed in DT40 cell assessed as calcium ion mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323704(CHEMBL1213158)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50194706(5'-deoxy-5'-benzyladenophostin A 2',3'',4''-trisph...)
Affinity DataEC50:  2.80nMAssay Description:Activity at rat IP3 type 1 receptor expressed in DT40 cell assessed as calcium ion mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at rat IP3R1 expressed in chicken DT40 cells assessed as induction of Ca2+ releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323708(CHEMBL1213161)
Affinity DataKd:  2.81nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50514587(CHEMBL4483666)
Affinity DataKd:  3.20nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50514587(CHEMBL4483666)
Affinity DataKd:  3.20nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184324(phosphoric acid mono-{(2R,3R,4R,5S,6R)-6-[(2S,3R,4...)
Affinity DataEC50:  4nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323710((1R,2R,3S,4R,6S)-3,6-dihydroxycyclohexane-1,2,4-tr...)
Affinity DataKd:  4.01nMAssay Description:Displacement of [3H]IP3 from rat recombinant N-terminal IP3R1 (1-604) expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184323(phosphoric acid mono-{(2R,3R,4R,5R,6R)-6-[(2R,3R,4...)
Affinity DataEC50:  4.60nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323705(CHEMBL1213159)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323707(CHEMBL1213160)
Affinity DataEC50:  5nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323706(CHEMBL1212943)
Affinity DataEC50:  5nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataKd:  7.60nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184325(2-[5-(6-amino-9H-9-purinyl)-2-hydroxymethyl-4-oxyp...)
Affinity DataKd:  7.60nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323709(CHEMBL1213163)
Affinity DataKd:  7.62nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50323708(CHEMBL1213161)
Affinity DataKd:  7.82nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  8.70nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  8.70nMAssay Description:Displacement of [3H]IP3 from rat IP3R1 expressed in human HEK cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  8.70nMAssay Description:Displacement of [3H]-IP3 from IP3R1 in Wistar rat cerebellar membrane measured after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50527899(CHEMBL4475041)
Affinity DataKd:  11nMAssay Description:Displacement of [3H]-IP3 from IP3R1 in Wistar rat cerebellar membrane measured after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50527899(CHEMBL4475041)
Affinity DataKd:  11nMAssay Description:Displacement of [3H]-IP3 from IP3R1 in Wistar rat cerebellar membrane measured after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Rat)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50184332(phosphoric acid mono-{(2R,3R,4R,5S,6R)-6-[(2S,3R,4...)
Affinity DataEC50:  11.3nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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