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TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.0410nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476140(CHEMBL373632)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85011(AcNH-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2018
Entry Details

TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85009(H2N-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50019568(CHEMBL411836 | SRIF-14 | Somatostatin receptor lig...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85012(AcNH-4-NO2-Phe-c[D-Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50592196(CHEMBL5174433)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at rat SST5More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50592196(CHEMBL5174433)
Affinity DataEC50:  0.316nMAssay Description:Agonist activity at rat SST5More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50592194(CHEMBL5195355)
Affinity DataEC50:  0.398nMAssay Description:Agonist activity at rat SST5More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50592194(CHEMBL5195355)
Affinity DataEC50:  0.398nMAssay Description:Agonist activity at rat SST5More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476137(CHEMBL222751)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2018
Entry Details

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214421(SOMATOSTATIN RECEPTOR LIGAND)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2018
Entry Details

TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | NSC_3086456 | MK 678)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  0.570nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476135(CHEMBL374316)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423340(CHEMBL250304)
Affinity DataKd:  0.741nMAssay Description:Displacement of [125I]SRIF14 from rat sst2 receptor from rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM405588(US10351547, Compound 2-2 | US10464918, Compound A ...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at rat SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50318385(2-(4-{[(2-{[(3-{[1-(5-{[(1R)-1-{[(4R,7S,10S,13R,16...)
Affinity DataIC50: 1.32nMAssay Description:Displacement of [111In]DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  1.43nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  1.47nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476143(CHEMBL376001)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82254(D-Nal-Cys-Tyr-D-Trp-Lys-Val-Cys-Thr-NH2 | DC-25-10...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  1.78nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50318388((4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-N-[(2R,3...)
Affinity DataIC50: 2.45nMAssay Description:Displacement of [111In]DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50318386(2-[7-({[2-({[3,5-bis({[1-(5-{[(1R)-1-{[(4R,7S,10S,...)
Affinity DataIC50: 2.45nMAssay Description:Displacement of [111In]DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85671(CAS_183658-72-2 | CYN 154806 | CYN-154806)
Affinity DataKi:  4.47nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50019568(CHEMBL411836 | SRIF-14 | Somatostatin receptor lig...)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85671(CAS_183658-72-2 | CYN 154806 | CYN-154806)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85013(H2N-4-NO2-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-N...)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50318387(CHEMBL1099306)
Affinity DataIC50: 14nMAssay Description:Displacement of [111In]DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85010(H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr...)
Affinity DataKi:  17.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476144(CHEMBL434761)
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85230(BIM 23313)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82257(D-Phe-Phe-Tyr-D-Trp-Lys-Val-Phe-Thr-NH2 | DC-25-12)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM85229(BIM 23295)
Affinity DataKi:  57nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  69nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  101nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  163nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM84629(BIM 23056)
Affinity DataKi:  835nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020202(CHEMBL2369466 | D-Tic-c(Cys-Tyr-D-Trp-Lys-Thr-Pen-...)
Affinity DataIC50: 949nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM82256(CAS_150155-61-6 | D-Phe-Phe-Tyr-D-Trp-Lys-Val-Phe-...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
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