Compile Data Set for Download or QSAR
Report error Found 52 for UniProtKB: P30988
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110268BDBM50110268(CSNLSTCVLGKLSQELc[DKLQK]YPRTNTGSGTP-amide | CHEMBL...)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024170BDBM50024170(CHEMBL2369912)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110272BDBM50110272(CSNLSTCVLGKLSQELc[DKLHK]YPRTNTGSGTP-amide | CHEMBL...)
Affinity DataKi:  0.0510nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639976BDBM50639976(Calcitonin (salmon synthetic) | Calcitonin salmon ...)
Affinity DataIC50: 0.0660nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110265BDBM50110265(CSNLSTCVLGKLSQELc[DKLHO]YPRTNTGSGTP-amide | CHEMBL...)
Affinity DataKi:  0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110275BDBM50110275(CGNLSTCBLGTYTQDF[DKFHO]YPQTAIGVGAP-amide | CHEMBL2...)
Affinity DataKi:  0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639976BDBM50639976(Calcitonin (salmon synthetic) | Calcitonin salmon ...)
Affinity DataIC50: 0.0890nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639983BDBM50639983(CHEMBL5567107)
Affinity DataIC50: 0.100nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639975BDBM50639975(Pramlintide | Pramlintida | Tripro-amylin | AC-013...)
Affinity DataIC50: 0.114nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639975BDBM50639975(Pramlintide | Pramlintida | Tripro-amylin | AC-013...)
Affinity DataIC50: 0.122nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639986BDBM50639986(CHEMBL5566450)
Affinity DataIC50: 0.213nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639990BDBM50639990(CHEMBL5554990)
Affinity DataIC50: 0.344nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639979BDBM50639979(CHEMBL5567446)
Affinity DataIC50: 0.355nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639988BDBM50639988(CHEMBL5560328)
Affinity DataIC50: 0.484nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110273BDBM50110273(CGNLSTCMLGTYTQDFc[DKFHK]FPQTAIGVGAP-amide | CHEMBL...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639992BDBM50639992(CHEMBL5567377)
Affinity DataIC50: 0.561nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639982BDBM50639982(CHEMBL5568431)
Affinity DataIC50: 0.589nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639987BDBM50639987(CHEMBL5568545)
Affinity DataIC50: 0.662nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639991BDBM50639991(CHEMBL5556440)
Affinity DataIC50: 0.745nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639985BDBM50639985(CHEMBL5561117)
Affinity DataIC50: 0.885nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639983BDBM50639983(CHEMBL5567107)
Affinity DataIC50: 1.09nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639978BDBM50639978(CHEMBL5568471)
Affinity DataIC50: 1.12nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639980BDBM50639980(CHEMBL5568414)
Affinity DataIC50: 1.13nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639981BDBM50639981(CHEMBL5568143)
Affinity DataIC50: 1.14nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639984BDBM50639984(CHEMBL5566453)
Affinity DataIC50: 1.14nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639975BDBM50639975(Pramlintide | Pramlintida | Tripro-amylin | AC-013...)
Affinity DataIC50: 1.49nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639989BDBM50639989(CHEMBL5560524)
Affinity DataIC50: 2.75nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639977BDBM50639977(CHEMBL5565993)
Affinity DataIC50: 5.09nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110267BDBM50110267(CGNLSTCBLGTYTQDFNKFHZYPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639980BDBM50639980(CHEMBL5568414)
Affinity DataIC50: 11.7nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639982BDBM50639982(CHEMBL5568431)
Affinity DataIC50: 11.9nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639988BDBM50639988(CHEMBL5560328)
Affinity DataIC50: 14.1nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639990BDBM50639990(CHEMBL5554990)
Affinity DataIC50: 15.5nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639987BDBM50639987(CHEMBL5568545)
Affinity DataIC50: 19.3nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639979BDBM50639979(CHEMBL5567446)
Affinity DataIC50: 19.5nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639986BDBM50639986(CHEMBL5566450)
Affinity DataIC50: 21.1nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639991BDBM50639991(CHEMBL5556440)
Affinity DataIC50: 22.9nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639978BDBM50639978(CHEMBL5568471)
Affinity DataIC50: 30.2nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639992BDBM50639992(CHEMBL5567377)
Affinity DataIC50: 42nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639985BDBM50639985(CHEMBL5561117)
Affinity DataIC50: 42.3nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110271BDBM50110271(CGNLSTCMLGTYTQDFNKFHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  43nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639989BDBM50639989(CHEMBL5560524)
Affinity DataIC50: 52.3nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639984BDBM50639984(CHEMBL5566453)
Affinity DataIC50: 73.4nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639977BDBM50639977(CHEMBL5565993)
Affinity DataIC50: 74.1nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCalcitonin receptor(Homo sapiens)
Novo Nordisk A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50639981BDBM50639981(CHEMBL5568143)
Affinity DataIC50: 102nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024171BDBM50024171(CHEMBL2369899)
Affinity DataKi:  195nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110266BDBM50110266(CGNLSTCMLGTYTQDFNKPHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  400nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422415BDBM50422415(CHEMBL2304022)
Affinity DataKi:  1.23E+3nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110276BDBM50110276(CGNLSTCMLGTYTQDFNPKHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIsoform 1 of Calcitonin receptor (1)(Human)
Rutgers University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110274BDBM50110274(CGNLSTCMLGTYTQDFNPGHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  2.57E+3nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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