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TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592204(CHEMBL5208674)
Affinity DataEC50:  0.0470nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592204(CHEMBL5208674)
Affinity DataEC50:  0.0501nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50051568(seglitide | CHEMBL311695 | (3S,6S,9S,12R,15S,18S)-...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50051568(seglitide | CHEMBL311695 | (3S,6S,9S,12R,15S,18S)-...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50051568(seglitide | CHEMBL311695 | (3S,6S,9S,12R,15S,18S)-...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50051568(seglitide | CHEMBL311695 | (3S,6S,9S,12R,15S,18S)-...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50051568(seglitide | CHEMBL311695 | (3S,6S,9S,12R,15S,18S)-...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataEC50:  0.0650nMAssay Description:Effective concentration on human somatostatin receptor 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592201(CHEMBL5179782)
Affinity DataEC50:  0.0710nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592201(CHEMBL5179782)
Affinity DataEC50:  0.0710nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592181(CHEMBL5178891)
Affinity DataEC50:  0.0770nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592181(CHEMBL5178891)
Affinity DataEC50:  0.0794nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM144757(US8952128, 15)
Affinity DataKi:  0.0800nM ΔG°:  -57.6kJ/molepH: 7.6 T: 2°CAssay Description:Membranes for in vitro receptor binding assays were obtained by the following procedures. CHO-K1 cells expressing one of the somatostatin receptors w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2015
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592185(CHEMBL5169724)
Affinity DataEC50:  0.0880nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50592185(CHEMBL5169724)
Affinity DataEC50:  0.0880nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM144752(US8952128, 11)
Affinity DataKi:  0.0900nM ΔG°:  -57.3kJ/molepH: 7.6 T: 2°CAssay Description:Membranes for in vitro receptor binding assays were obtained by the following procedures. CHO-K1 cells expressing one of the somatostatin receptors w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2015
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474235(CHEMBL3349606)
Affinity DataKi:  0.100nMAssay Description:Binding affinity towards human Somatostatin receptor type 5 (sst5) using Tyr11-[125I]-SRIF as radioligand was determined in COS cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50468144(CHEMBL4286244)
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at human SSR5 expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 15 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474236(CHEBI:72312 | CHEMBL3349607)
Affinity DataKi:  0.126nMAssay Description:Binding affinity towards human Somatostatin receptor type 5 (sst5) using Tyr11-[125I]-SRIF as radioligand was determined in COS cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM123235(US8742110, 3-20)
Affinity DataIC50: 0.129nMpH: 7.8Assay Description:SSTR5 binding assays can be performed by labeling somatostatin and determining the ability of a compound to inhibit somatostatin binding. (Poitout et...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2014
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.140nMAssay Description:Inhibition of human sst5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM123247(US8742110, 4-11)
Affinity DataIC50: 0.152nMpH: 7.8Assay Description:SSTR5 binding assays can be performed by labeling somatostatin and determining the ability of a compound to inhibit somatostatin binding. (Poitout et...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2014
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474221(CHEMBL3349521)
Affinity DataKi:  0.158nMAssay Description:Binding affinity towards human Somatostatin receptor type 5 (sst5) using Tyr11-[125I]-SRIF as radioligand was determined in COS cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM144751(US8952128, 10)
Affinity DataKi:  0.160nM ΔG°:  -55.9kJ/molepH: 7.6 T: 2°CAssay Description:Membranes for in vitro receptor binding assays were obtained by the following procedures. CHO-K1 cells expressing one of the somatostatin receptors w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2015
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85247(Tyr10-cortistatin)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85560(CST14-Tyr10)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM123253(US8742110, 4-17)
Affinity DataIC50: 0.165nMpH: 7.8Assay Description:SSTR5 binding assays can be performed by labeling somatostatin and determining the ability of a compound to inhibit somatostatin binding. (Poitout et...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2014
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM123270(US8742110, 5-6)
Affinity DataIC50: 0.172nMpH: 7.8Assay Description:SSTR5 binding assays can be performed by labeling somatostatin and determining the ability of a compound to inhibit somatostatin binding. (Poitout et...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2014
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM123248(US8742110, 4-12)
Affinity DataIC50: 0.188nMpH: 7.8Assay Description:SSTR5 binding assays can be performed by labeling somatostatin and determining the ability of a compound to inhibit somatostatin binding. (Poitout et...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2014
Entry Details
US Patent

TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85323(LTT-SRIF28 | SRIF28-Leu8,D-Trp22,Tyr25)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataEC50:  0.190nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84989(SS-25)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85323(LTT-SRIF28 | SRIF28-Leu8,D-Trp22,Tyr25)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
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