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Found 23 for UniProtKB: P53610
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM14459((+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of rat brain GGTase1 assessed as decrease in transfer of [3H]H]geranylgeranyl from [3H]geranylgeranyl PPi to H-Ras-CVLL after 30 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481906(CHEMBL1075839)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50075437(2,4,5-Trifluoro-6-nitro-3-((2E,6E)-3,7,11-trimethy...)
Affinity DataIC50:  1.25E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481911(CHEMBL1075809)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481907(CHEMBL1075810)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481909(CHEMBL1075863)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075439(3-Benzyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMB...)
Affinity DataIC50:  5.80E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075440(2,4,5-Trifluoro-3-(4-isopropenyl-cyclohex-1-enylme...)
Affinity DataIC50:  8.50E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481908(CHEMBL1075861)
Affinity DataIC50:  9.80E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481910(CHEMBL1075859)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481912(CHEMBL1075865)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50075443(3-Dodecyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504717(CHEMBL4459281)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504718(CHEMBL4564870)
Affinity DataIC50:  1.45E+5nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50075442(3-Allyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMBL...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075438(3-(Biphenyl-4-ylmethoxy)-2,4,5-trifluoro-6-nitro-p...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075441(2,4,5-Trifluoro-3-(naphthalen-2-ylmethoxy)-6-nitro...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504716(CHEMBL4589567)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50273716(CHEMBL457423 | [2-(Benzoimidazol-1-yl)ethyl]-bisph...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504719(CHEMBL4438314)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504720(CHEMBL4529809)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504715(CHEMBL4514446)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504714(CHEMBL4460301)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed