Compile Data Set for Download or QSAR
Report error Found 23 for UniProtKB: P53610
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 14459BDBM14459((+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat brain GGTase1 assessed as decrease in transfer of [3H]H]geranylgeranyl from [3H]geranylgeranyl PPi to H-Ras-CVLL after 30 mins by l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481906BDBM50481906(CHEMBL1075839)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075437BDBM50075437(2,4,5-Trifluoro-6-nitro-3-((2E,6E)-3,7,11-trimethy...)
Affinity DataIC50: 1.25E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481911BDBM50481911(CHEMBL1075809)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481907BDBM50481907(CHEMBL1075810)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481909BDBM50481909(CHEMBL1075863)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075439BDBM50075439(3-Benzyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMB...)
Affinity DataIC50: 5.80E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075440BDBM50075440(2,4,5-Trifluoro-3-(4-isopropenyl-cyclohex-1-enylme...)
Affinity DataIC50: 8.50E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481908BDBM50481908(CHEMBL1075861)
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481910BDBM50481910(CHEMBL1075859)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075443BDBM50075443(3-Dodecyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481912BDBM50481912(CHEMBL1075865)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504717BDBM50504717(CHEMBL4459281)
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504718BDBM50504718(CHEMBL4564870)
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075441BDBM50075441(2,4,5-Trifluoro-3-(naphthalen-2-ylmethoxy)-6-nitro...)
Affinity DataIC50: 2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075438BDBM50075438(3-(Biphenyl-4-ylmethoxy)-2,4,5-trifluoro-6-nitro-p...)
Affinity DataIC50: 2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50075442BDBM50075442(3-Allyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMBL...)
Affinity DataIC50: 2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504716BDBM50504716(CHEMBL4589567)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504714BDBM50504714(CHEMBL4460301)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504719BDBM50504719(CHEMBL4438314)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504720BDBM50504720(CHEMBL4529809)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273716BDBM50273716([2-(Benzoimidazol-1-yl)ethyl]-bisphosphonic acid |...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rat)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504715BDBM50504715(CHEMBL4514446)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed