Compile Data Set for Download or QSAR
maximum 50k data
Found 58 of affinity data for UniProtKB/TrEMBL: P54652
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKi: >200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531168(CHEMBL4525506)
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531168(CHEMBL4525506)
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKi: >200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi:  220nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.33 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi:  220nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.33 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  250nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 2 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  250nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 2 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  520nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  520nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531171(CHEMBL4556409)
Affinity DataKi:  1.40E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 24 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531171(CHEMBL4556409)
Affinity DataKi:  1.40E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 24 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531171(CHEMBL4556409)
Affinity DataKi:  2.00E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 2 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531171(CHEMBL4556409)
Affinity DataKi:  2.00E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 2 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531171(CHEMBL4556409)
Affinity DataKi:  2.50E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531171(CHEMBL4556409)
Affinity DataKi:  2.50E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi:  3.30E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi:  3.30E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531170(CHEMBL4593659)
Affinity DataKi:  3.50E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531170(CHEMBL4593659)
Affinity DataKi:  3.50E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531170(CHEMBL4593659)
Affinity DataKi:  3.55E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531170(CHEMBL4593659)
Affinity DataKi:  3.55E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  3.70E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 46 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  3.70E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 46 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi:  4.70E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531165(CHEMBL4519613)
Affinity DataKi:  4.70E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  6.90E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  6.90E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  7.20E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 19 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  7.20E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 19 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531172(CHEMBL4452822)
Affinity DataKi:  8.00E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531172(CHEMBL4452822)
Affinity DataKi:  8.00E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  1.00E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531166(CHEMBL4545529)
Affinity DataKi:  1.00E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531172(CHEMBL4452822)
Affinity DataKi:  1.20E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.33 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531172(CHEMBL4452822)
Affinity DataKi:  1.20E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.33 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  1.70E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  1.70E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  1.80E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531167(CHEMBL4583945)
Affinity DataKi:  1.80E+4nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531172(CHEMBL4452822)
Affinity DataKi:  1.10E+5nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531172(CHEMBL4452822)
Affinity DataKi:  1.10E+5nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531169(CHEMBL4592795)
Affinity DataKi: >2.00E+5nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531169(CHEMBL4592795)
Affinity DataKi: >2.00E+5nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531169(CHEMBL4592795)
Affinity DataKi: >2.00E+5nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 2 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50531169(CHEMBL4592795)
Affinity DataKi: >2.00E+5nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 2 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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