Compile Data Set for Download or QSAR
Report error Found 9 of affinity data for UniProtKB/TrEMBL: P68371
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  1.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  2.68E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataKd:  223nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50410800(CHEMBL5206193)
Affinity DataIC50: 108nMAssay Description:Inhibition of beta-tubulin polymerization (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50475439(CHEMBL383775)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against tubulin using tubulin polymerization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50410801(CHEMBL5276251)
Affinity DataIC50: 5.51E+3nMAssay Description:Inhibition of beta-tubulin polymerization (unknown origin) measured every 3 secs for 1 hr by spectrofluorometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50594719(CHEMBL5186583)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of beta-tubulin polymerization in human HCT-116 cells using TMB substrate by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTubulin beta-4B chain(Human)TBA
LigandPNGBDBM50475438(CHEMBL364477)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity against tubulin using tubulin polymerization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed