TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Antagonist activity at full length ERbeta (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucifer...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.60nMAssay Description:Antagonist activity at full length ERbeta (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucifer...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.70nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 2.60nMAssay Description:Antagonist activity at full length ERbeta (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucifer...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 2.70nMAssay Description:Antagonist activity at full length ERbeta (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucifer...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 2.90nMAssay Description:Antagonist activity at full length ERalpha (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucife...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Binding affinity to full length human His-tagged ROR1 (937 residues ) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 4nMAssay Description:Antagonist activity at full length ERbeta (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucifer...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 4.10nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 6.70nMAssay Description:Antagonist activity at full length ERalpha (unknown origin) assessed as reduction in E2 induced response after 24 hrs by cell based ERE-driven lucife...More data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 7.10nMAssay Description:Agonist activity at full length ERbeta (unknown origin) after 24 hrs by cell based ERE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.90nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding affinity to full length human His-tagged ROR1 (937 residues ) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Binding affinity to human ROR1 expressed in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 22nMAssay Description:Binding affinity to full length human His-tagged ROR1 (937 residues ) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 34nMAssay Description:Binding affinity to full length human His-tagged ROR1 (937 residues ) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Binding affinity to ROR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 160nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 180nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 260nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetInactive tyrosine-protein kinase transmembrane receptor ROR1(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 330nMAssay Description:Binding affinity to ROR1 kinase domain (453 to 783 residues) (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair












































