TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of Cysteine protease falcipain-3 in Plasmodium falciparum HB3 infected erythrocytes by Z-Phe-Arg-AMC substrate hydrolysis assayMore data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of Cysteine protease falcipain-3 in Plasmodium falciparum HB3-leuR1 mutant infected erythrocytes by Z-Phe-Arg-AMC substrate hydrolysis ass...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 407nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 459nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 482nMAssay Description:Inhibition of Plasmodium falciparum falcipain 3 incubated with compound for 10 mins before addition of 25 uM Z-Leu-Arg-AMC substrate by fluorescence ...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 484nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 547nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 851nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 8.22E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 8.56E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-3 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins ...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 8.79E+3nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 9.98E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-3 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins ...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair