Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of affinity data for UniProtKB/TrEMBL: Q8IYL9
TargetPsychosine receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175290(CHEMBL3810385)
Affinity DataIC50: >1.00E+4nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged TDAG8 receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP res...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPsychosine receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM123510(US8748435, 35)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of TDAG8 (unknown origin) expressed in human HeLa cells assessed as reduction in cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPsychosine receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50260351(CHEMBL4086667)
Affinity DataIC50: >2.30E+4nMAssay Description:Antagonist activity at human TDAG8 expressed in human HeLa cells assessed as inhibition of IBMX-induced cAMP accumulation preincubated for 10 mins fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPsychosine receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50260350(CHEMBL4078089)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human TDAG8 expressed in human HeLa cells assessed as inhibition of IBMX-induced cAMP accumulation preincubated for 10 mins fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed