TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of human NEK9 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of human NEK9 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human NEK9 (1 to 324 residues) using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human NEK9 using MBP as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human NEK9 (1 to 324 residues) using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human GST-tagged NEK9 catalytic domain (347 to 732 residues) expressed in baculovirus expression system using serine/threon...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 9.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 3.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 6.70E+3nMAssay Description:Average Binding Constant for NEK9; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 5.40E+3nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 3.10E+3nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 3.10E+3nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK9More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 790nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek9(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK9 kinase domainMore data for this Ligand-Target Pair