Compile Data Set for Download or QSAR
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Found 10 of affinity data for UniProtKB/TrEMBL: Q99986
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50:  33nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50502749(CHEMBL4435359)
Affinity DataIC50:  150nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50502748(CHEMBL4436323)
Affinity DataIC50:  260nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50502751(CHEMBL4452098)
Affinity DataIC50:  674nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  743nMAssay Description:Inhibition of human VRK1 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human VRK1 using [KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK] as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human VRK1 in presence of 10 uM ATP by radiometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50001733(CHEMBL3133821)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human VRK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50331612(CHEMBL1290072 | N-(4-methoxybenzyl)benzofuro[2,3-b...)
Affinity DataIC50:  1.29E+5nMAssay Description:Inhibition of human VRK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)

Curated by ChEMBL
LigandPNGBDBM50502749(CHEMBL4435359)
Affinity DataKd:  190nMAssay Description:Binding affinity to recombinant full length N-terminal His-tagged VRK1 (unknown origin) (1 to 396 residues) expressed in Escherichia coli BL 21 DE3-R...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed