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Report error Found 2918 for UniProtKB: Q9UDY8
LigandChemical structure of BindingDB Monomer ID 355969BDBM355969(US9815842, Example 93 | (S)-1-(5-chloro-6- (difluo...)
Affinity DataIC50: 0.00100nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355969BDBM355969(US9815842, Example 93 | (S)-1-(5-chloro-6- (difluo...)
Affinity DataIC50: 0.00100nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355980BDBM355980(US9815842, Example 104 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355967BDBM355967(US9815842, Example 91 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50169049BDBM50169049(CHEMBL3806155 | US9815842, Example 1 | US10442808,...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50169049BDBM50169049(CHEMBL3806155 | US9815842, Example 1 | US10442808,...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355970BDBM355970(US9815842, Example 94 | (S)-1-(6-(2H-1,2,3- triazo...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355971BDBM355971(US9815842, Example 95 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355970BDBM355970(US9815842, Example 94 | (S)-1-(6-(2H-1,2,3- triazo...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50169049BDBM50169049(CHEMBL3806155 | US9815842, Example 1 | US10442808,...)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of MALT1 C domain (329 to 824 residues) (unknown origin) using Ac-Trp-Leu-Arg-Ser-Arg-Cys(PT14)-NH2 as substrate preincubated for 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 355971BDBM355971(US9815842, Example 95 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355967BDBM355967(US9815842, Example 91 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355889BDBM355889(US9815842, Example 13 | (S)-methyl 3-chloro- 5-(3-...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355886BDBM355886(US9815842, Example 10 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355950BDBM355950(US9815842, Example 74 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355892BDBM355892(US9815842, Example 16 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355889BDBM355889(US9815842, Example 13 | (S)-methyl 3-chloro- 5-(3-...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355892BDBM355892(US9815842, Example 16 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355885BDBM355885(US9815842, Example 9 | (S)-1-(5-chloro-6- methoxyp...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355980BDBM355980(US9815842, Example 104 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355886BDBM355886(US9815842, Example 10 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355950BDBM355950(US9815842, Example 74 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355885BDBM355885(US9815842, Example 9 | (S)-1-(5-chloro-6- methoxyp...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355948BDBM355948(US9815842, Example 72 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355897BDBM355897(US9815842, Example 21 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355894BDBM355894(US9815842, Example 18 | 1-(5-chloro-6- methoxypyri...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355895BDBM355895(US9815842, Example 19 | 1-(2-chloro-7- isopropylpy...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355890BDBM355890(US9815842, Example 14 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355896BDBM355896(US9815842, Example 20 | 1-(3-chloro-4-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355890BDBM355890(US9815842, Example 14 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355948BDBM355948(US9815842, Example 72 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355978BDBM355978(US9815842, Example 102 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355915BDBM355915(US9815842, Example 39 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355973BDBM355973(US9815842, Example 97 | (S)-1-(5-chloro-6- (difluo...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355973BDBM355973(US9815842, Example 97 | (S)-1-(5-chloro-6- (difluo...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355911BDBM355911(US9815842, Example 35 | 1-(7-(sec-butyl)-2- chloro...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355906BDBM355906(US9815842, Example 30 | 1-(2-chloro-7- isopropylpy...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355896BDBM355896(US9815842, Example 20 | 1-(3-chloro-4-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355906BDBM355906(US9815842, Example 30 | 1-(2-chloro-7- isopropylpy...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355897BDBM355897(US9815842, Example 21 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355894BDBM355894(US9815842, Example 18 | 1-(5-chloro-6- methoxypyri...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355895BDBM355895(US9815842, Example 19 | 1-(2-chloro-7- isopropylpy...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355965BDBM355965(US9815842, Example 89 | (S)-1-(2-chloro-7-(1- meth...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355965BDBM355965(US9815842, Example 89 | (S)-1-(2-chloro-7-(1- meth...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355921BDBM355921(US9815842, Example 45 | (R)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355925BDBM355925(US9815842, Example 49 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355925BDBM355925(US9815842, Example 49 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355987BDBM355987(US9815842, Example 111 | (R)-1-(6-(2H-1,2,3- triaz...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355921BDBM355921(US9815842, Example 45 | (R)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355987BDBM355987(US9815842, Example 111 | (R)-1-(6-(2H-1,2,3- triaz...)
Affinity DataIC50: 0.00300nMAssay Description:The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details
US Patent

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