Compile Data Set for Download or QSAR
Report error Found 127 of affinity data for UniProtKB/TrEMBL: Q9ULZ1
TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610889(US10626096, Example 2 | 2-({[4-(2,6-Dimethoxypheny...)
Affinity DataEC50:  1nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610890(US10626096, Example 3 | 7-Chloro-2-({[4-(2,6-dimet...)
Affinity DataEC50:  2nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610898(US10626096, Example 11 | [2-({[4-(2,6-Dimethoxyphe...)
Affinity DataEC50:  5nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610988(US10626096, Example 95 | 2-{[4-(2,6-Dimethoxypheny...)
Affinity DataEC50:  6nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610925(US10626096, Example 38 | {[4-(2,6-Dimethoxyphenyl)...)
Affinity DataEC50:  9nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610922(US10626096, Example 35)
Affinity DataEC50:  10nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610926(US10626096, Example 39)
Affinity DataEC50:  11nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610929(US10626096, Example 42)
Affinity DataEC50:  12nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610896(US10626096, Example 9 | (2E)-3-[4-(2,6-Dimethoxyph...)
Affinity DataEC50:  18nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610935(US10626096, Example 48 | 4-[4-(2,6-Dimethoxyphenyl...)
Affinity DataEC50:  22nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610892(US10626096, Example 5 | {[4-(2,6-Dimethoxyphenyl)-...)
Affinity DataEC50:  26nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610888(US10626096, Example 1 | 4-(2,6-Dimethoxyphenyl)-5-...)
Affinity DataEC50:  31nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610967(US10626096, Example 78 | 2-({[4-(2,6-Dimethoxyphen...)
Affinity DataEC50:  34nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610977(US10626096, Example 88 | {[4-(2,6-Dimethoxyphenyl)...)
Affinity DataEC50:  35nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610930(US10626096, Example 43)
Affinity DataEC50:  39nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610928(US10626096, Example 41)
Affinity DataEC50:  45nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610998(US10626096, Example 103)
Affinity DataEC50:  46nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610943(US10626096, Example 56 | (2Z)-3-[4-(2,6-Dimethoxyp...)
Affinity DataEC50:  48nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610999(US10626096, Example 104 | 5-({[4-(2,6-Dimethoxyphe...)
Affinity DataEC50:  48nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610951(US10626096, Example 64 | (2E)-3-[4-(2,6-dimethoxyp...)
Affinity DataEC50:  52nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610913(US10626096, Example 26)
Affinity DataEC50:  57nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610970(US10626096, Example 81 | Methyl 4-({[4-(2,6-dimeth...)
Affinity DataEC50:  71nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610987(US10626096, Example 94 | 3-({[4-(2,6-Dimethoxyphen...)
Affinity DataEC50:  71nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610952(US10626096, Example 65 | (2E)-3-[4-(2,6-dimethoxyp...)
Affinity DataEC50:  75nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610909(US10626096, Example 22)
Affinity DataEC50:  87nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009560(CHEMBL3234454)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610960(US10626096, Example 72 | N-{[4-(2,6-Dimethoxypheny...)
Affinity DataEC50:  95nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
Go to US Patent

TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610933(US10626096, Example 46 | 3-[4-(2,6-Dimethoxyphenyl...)
Affinity DataEC50:  96nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610962(US10626096, Example 74)
Affinity DataEC50:  98nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610997(US10626096, Example 102 | ({[4-(2,6-Dimethoxypheny...)
Affinity DataEC50:  103nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610923(US10626096, Example 36)
Affinity DataEC50:  108nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610938(US10626096, Example 51 | Ethyl (3E)-4-[4-(2,6-dime...)
Affinity DataEC50:  111nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610891(US10626096, Example 4 | Ethyl {[4-(2,6-dimethoxyph...)
Affinity DataEC50:  122nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610963(US10626096, Example 75 | 3-({[4-(2,6-Dimethoxyphen...)
Affinity DataEC50:  128nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610921(US10626096, Example 34)
Affinity DataEC50:  152nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610964(US10626096, Example 76 | 4-(2,6-Dimethoxyphenyl)-3...)
Affinity DataEC50:  158nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610900(US10626096, Example 13 | 3-[4-(2,6-Dimethoxyphenyl...)
Affinity DataEC50:  159nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610902(US10626096, Example 15 | 6-({[4-(2,6-Dimethoxyphen...)
Affinity DataEC50:  164nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610981(US10626096, Example 92 | (4R)-1-{(2E)-3-[4-(2,6-Di...)
Affinity DataEC50:  166nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610906(US10626096, Example 19 | (2E)-3-[4-(2,6-Dimethoxyp...)
Affinity DataEC50:  171nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610918(US10626096, Example 31)
Affinity DataEC50:  174nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009571(CHEMBL3234461)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610897(US10626096, Example 10)
Affinity DataEC50:  192nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610968(US10626096, Example 79 | Methyl 3-({[4-(2,6-dimeth...)
Affinity DataEC50:  208nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610939(US10626096, Example 52 | 2-{(E)-2-[4-(2,6-Dimethox...)
Affinity DataEC50:  217nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610972(US10626096, Example 83 | 2-{[4-(2,6-Dimethoxypheny...)
Affinity DataEC50:  219nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610974(US10626096, Example 85 | 4-(2,6-Dimethoxyphenyl)-3...)
Affinity DataEC50:  253nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610978(US10626096, Example 89 | Methyl {[4-(2,6-dimethoxy...)
Affinity DataEC50:  261nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM610973(US10626096, Example 84 | {[4-(2,6-Dimethoxyphenyl)...)
Affinity DataEC50:  267nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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