Compile Data Set for Download or QSAR
Report error Found 345 for UniProtKB: Q9WUD2
LigandPNGBDBM50222640(CHEMBL415543)
Affinity DataIC50: 0.320nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222640(CHEMBL415543)
Affinity DataIC50: 0.320nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222695(CHEMBL155433)
Affinity DataIC50: 0.460nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222637(CHEMBL154743)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222696(CHEMBL156041)
Affinity DataIC50: 0.550nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222635(CHEMBL267205)
Affinity DataIC50: 0.720nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222647(CHEMBL154990)
Affinity DataIC50: 0.950nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222649(CHEMBL155730)
Affinity DataIC50: 0.950nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222641(CHEMBL157962)
Affinity DataIC50: 1.20nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222638(CHEMBL422702)
Affinity DataIC50: 2.40nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222644(CHEMBL434295)
Affinity DataIC50: 2.5nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222648(CHEMBL156693)
Affinity DataIC50: 3nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222639(CHEMBL356682)
Affinity DataIC50: 3.20nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222646(CHEMBL157917)
Affinity DataIC50: 5.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222694(CHEMBL158189)
Affinity DataIC50: 6.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222691(CHEMBL156927)
Affinity DataIC50: 9.30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222690(CHEMBL345157)
Affinity DataIC50: 10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222645(CHEMBL157918)
Affinity DataIC50: 11nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222693(CHEMBL157579)
Affinity DataIC50: 12nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50224228(CHEMBL46233)
Affinity DataIC50: 15nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224175(CHEMBL48061)
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224176(CHEMBL296963)
Affinity DataIC50: 30nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50222689(CHEMBL157774)
Affinity DataEC50: >30nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222636(CHEMBL155978)
Affinity DataEC50: >30nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222634(CHEMBL157473)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222692(CHEMBL348634)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  30nMAssay Description:In vitro agonist activity, increased [Ca2+] influx, at vanilloid receptor of rat dorsal root gangliaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50222643(CHEMBL157688)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM20321(JYL1421 | CHEMBL388824 | 3-[(4-tert-butylphenyl)me...)
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM20321(JYL1421 | CHEMBL388824 | 3-[(4-tert-butylphenyl)me...)
Affinity DataIC50: 37nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
LigandPNGBDBM50470963(CHEMBL146728)
Affinity DataEC50:  41nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandPNGBDBM50470958(CHEMBL60744)
Affinity DataEC50:  56nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandPNGBDBM50231166(CHEMBL58719)
Affinity DataEC50:  60nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
LigandPNGBDBM50224232(CHEMBL296729)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224234(CHEMBL45252)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224229(CHEMBL48998)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50231166(CHEMBL58719)
Affinity DataEC50:  60nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
LigandPNGBDBM50224196(CHEMBL43723)
Affinity DataIC50: 66nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224237(CHEMBL431341)
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224230(CHEMBL47282)
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50470962(CHEMBL144805)
Affinity DataEC50:  75nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandPNGBDBM50231204(CHEMBL80662)
Affinity DataEC50:  100nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
LigandPNGBDBM161012(US9108905, 1 | US9186360, 89)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293F cells assessed as inhibition of 2APB-induced increase in intracellular Ca2+ level by FLIPR-base...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50231186(CHEMBL309891)
Affinity DataEC50:  110nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50463972(CHEMBL4249976)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50470976(CHEMBL146099)
Affinity DataEC50:  130nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandPNGBDBM50470956(CHEMBL424317)
Affinity DataEC50:  130nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 345 total ) | Next | Last >>
Jump to: