TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.90E+4nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 3.10E+3nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 5.80E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 8.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 7.03E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 56nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 510nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 3.52E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 75nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 5.48E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 5.13E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 1.66E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 330nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 2.72E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 5.30E+4nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 5.48E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 710nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 6.14E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 1.34E+3nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at rat TRPV2 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >30nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >30nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research
Curated by ChEMBL
Sandoz Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair






























3D Structure (crystal)

















