TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant wild-type PAD2 (unknown origin) using N-alpha-Benzoyl-L-arginine ethyl ester as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant wild-type PAD2 (unknown origin) using N-alpha-Benzoyl-L-arginine ethyl ester as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of recombinant wild-type PAD2 (unknown origin) using N-alpha-Benzoyl-L-arginine ethyl ester as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of recombinant wild-type PAD2 (unknown origin) using N-alpha-Benzoyl-L-arginine ethyl ester as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 5.90E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Irreversible inhibition of PAD2 assessed as hydrolysis of benzoyl-L-arginine ethyl ester preincubated for 15 mins measured after 15 mins by fluoromet...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataIC50: 6.32E+3nMAssay Description:Inhibition of recombinant wild-type PAD2 (unknown origin) using N-alpha-Benzoyl-L-arginine ethyl ester as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 7.50E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 7.60E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataKi: 8.08E+3nMAssay Description:Inhibition of recombinant wild-type PAD2 (unknown origin) using N-alpha-Benzoyl-L-arginine ethyl ester as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 8.30E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
Affinity DataEC50: 9.50E+3nMAssay Description:Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu...More data for this Ligand-Target Pair
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL
TargetProtein-arginine deiminase type-2(Human)
The Scripps Research Institute-Florida
Curated by ChEMBL
The Scripps Research Institute-Florida
Curated by ChEMBL











































