BDBM50000310 6-(2-Imidazol-1-yl-vinyl)-3,4-dihydro-1H-quinolin-2-one::CHEMBL160790

SMILES O=C1CCc2cc(\C=C\n3ccnc3)ccc2N1

InChI Key InChIKey=PERHUGCCUROAON-FNORWQNLSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50000310   

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000310(6-(2-Imidazol-1-yl-vinyl)-3,4-dihydro-1H-quinolin-...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human blood platelet c-AMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000310(6-(2-Imidazol-1-yl-vinyl)-3,4-dihydro-1H-quinolin-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Compound was evaluated for the inhibition of human blood platelet thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed