TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0210nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0310nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0470nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: >300nMAssay Description:Partial agonist activity at rat alpha6 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Homo sapiens (Human))
Boise State University
Curated by ChEMBL
Boise State University
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Homo sapiens (Human))
Boise State University
Curated by ChEMBL
Boise State University
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Homo sapiens (Human))
Boise State University
Curated by ChEMBL
Boise State University
Curated by ChEMBL
Affinity DataIC50: 0.390nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Homo sapiens (Human))
Boise State University
Curated by ChEMBL
Boise State University
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at nAChRalpha6beta2 in Sprague-Dawley rat striatal slices assessed as inhibition of nicotine-evoked [3H]dopamine uptake by liquid...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Homo sapiens (Human))
Boise State University
Curated by ChEMBL
Boise State University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.22nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 8.59nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 9.91nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 37.4nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Homo sapiens (Human))
Boise State University
Curated by ChEMBL
Boise State University
Curated by ChEMBL
Affinity DataIC50: 201nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 205nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 222nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair