BDBM50263131 (+)-7-Methyl-2-exo-[3'-(6-fluoropyridin-2-yl)-5'-pyridinyl]-7-azabicyclo[2.2.1]heptane::(-)-7-Methyl-2-exo-[3'-(6-fluoropyridin-2-yl)-5'-pyridinyl]-7-azabicyclo[2.2.1]heptane::CHEMBL478447
SMILES CN1[C@@H]2CC[C@@H]1[C@H](C2)c1cncc(c1)-c1cccc(F)n1
InChI Key InChIKey=JGOKWXDQJRLPLM-IIAWOOMASA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50263131
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKd: 0.540nMAssay Description:Binding affinity to human alpha4beta2 nAChR expressed in human SHEP1 cellsMore data for this Ligand-Target Pair