Affinity DataKi: 0.950nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by ChEMBL
University Of Texas Medical Branch
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]-SCH23390 from wild type human D1R expressed in HEK293 cell membranes incubated for 90 mins by scintillation counting based compe...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Compound was evaluated for its ability to displace [3H]WIN-35428 binding in rat caudate-putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Compound was evaluated for its ability to displace [3H]WIN-35428 binding in rat caudate-putamenMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by ChEMBL
University Of Texas Medical Branch
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-SCH23390 from wild type human D1R expressed in HEK293 cell membranes incubated for 90 mins by scintillation counting based compe...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Compound was evaluated for its ability to displace [3H]WIN-35428 binding in rat caudate-putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 30nM ΔG°: -42.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 30nM ΔG°: -42.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 30nM ΔG°: -42.9kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Compound was evaluated for its ability to displace [3H]WIN-35428 binding in rat caudate-putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 40nM ΔG°: -42.2kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]pirenzepine displacement.More data for this Ligand-Target Pair