Affinity DataKi: 0.174nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.275nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.692nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 26nMpH: 5.2Assay Description:Competitive inhibition of human recombinant beta-glucocerebrosidase assessed as 4-methyumbelliferone formation after 30 mins by Lineweaver-Burk plot ...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 60nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 80nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 90nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 170nMpH: 5.2Assay Description:Competitive inhibition of human recombinant beta-glucocerebrosidase assessed as 4-methyumbelliferone formation after 30 mins by Lineweaver-Burk plot ...More data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMpH: 5.2Assay Description:Competitive inhibition of human recombinant beta-glucocerebrosidase assessed as 4-methyumbelliferone formation after 30 mins by Lineweaver-Burk plot ...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 330nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 479nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 700nMpH: 5.2Assay Description:Competitive inhibition of human recombinant beta-glucocerebrosidase assessed as 4-methyumbelliferone formation after 30 mins by Lineweaver-Burk plot ...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 770nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 820nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 820nMAssay Description:Binding affinity to recombinant imiglucerase using 4-methylumbelliferyl-beta-D-glucopyranoside as substrate preincubated for 30 mins before substrate...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 890nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair