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Found 4 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A' and Ligand = 'BDBM50598931'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataKi:  1.80nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataKi:  35nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataEC50:  0.447nMAssay Description:Agonist activity at human melatonin MT1 receptor stably expressing in human HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataEC50:  0.589nMAssay Description:Agonist activity at human melatonin MT1 receptor stably expressing in human HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed