Affinity DataKi: 0.0100nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity of the [35S]- radiolabelled compound to rhesus monkey Bradykinin receptor B1More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity of the [35S]- radiolabelled compound to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo rec...More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity of the [35S]- radiolabelled compound to rabbit Bradykinin receptor B1More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity of the [35S]- radiolabelled compound to dog Bradykinin receptor B1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.09nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.73nMAssay Description:Binding affinity to human Bradykinin receptor B1 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24.5nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity of the [35S]- radiolabelled compound to rat Bradykinin receptor B1More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.65E+3nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the [35S]- radiolabelled compound to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo rec...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Bradykinin receptor B2 over-expressed in transgenic rats was determined by ex vivo receptor occupancy assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Antagonist activity of the compound against human Bradykinin receptor B1 was determined in a fluorescence imaging plate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Antagonist activity in human bradykinin B1 receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Antagonist activity in human bradykinin B1 receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataKd: 0.0150nMAssay Description:Equilibrium dissociation constant of the [35S]- radiolabelled compound against human Bradykinin receptor B1 expressed in CHO membranes was determinedMore data for this Ligand-Target Pair