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Found 68 with Last Name = 'tahara' and Initial = 't'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452985(CHEMBL2114234)
Affinity DataKi:  6.70nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452983(CHEMBL2114236)
Affinity DataKi:  9.40nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452981(CHEMBL2115231)
Affinity DataKi:  9.60nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452980(CHEMBL2115232)
Affinity DataKi:  21nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452984(CHEMBL2114235)
Affinity DataKi:  23nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM81774(CAS_15676-16-1 | SULPIRIDE,(+) | Sulpiride-S | Sul...)
Affinity DataKi:  29nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50284586(CHEMBL22857 | N-((S)-1-Butyl-pyrrolidin-2-ylmethyl...)
Affinity DataKi:  51nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452990(CHEMBL2114240)
Affinity DataKi:  59nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452982(CHEMBL2115229)
Affinity DataKi:  95nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452987(CHEMBL2115228)
Affinity DataKi:  210nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50284609(CHEMBL278762 | N-((R)-1-Butyl-pyrrolidin-2-ylmethy...)
Affinity DataKi:  230nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452988(CHEMBL2114238)
Affinity DataKi:  400nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452986(CHEMBL2115227)
Affinity DataKi:  630nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452989(CHEMBL2114239)
Affinity DataKi:  650nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452979(CHEMBL2115233)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM81775(Sulpiride-R | Sulpiride-d | Sulpiride-high,(-) | S...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  28nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460520(CHEMBL4228293)
Affinity DataIC50:  44nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460521(CHEMBL4228332)
Affinity DataIC50:  51nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460518(CHEMBL4228977)
Affinity DataIC50:  81nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460523(CHEMBL4225627)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460524(CHEMBL4225893)
Affinity DataIC50:  560nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460522(CHEMBL4226829)
Affinity DataIC50:  590nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460518(CHEMBL4228977)
Affinity DataIC50:  590nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460521(CHEMBL4228332)
Affinity DataIC50:  730nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460523(CHEMBL4225627)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50366597(2-Acetylfuranonaphthoquinone | BBI-608 | Napabucas...)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of IL-6 induced STAT3 phosphorylation at Tyr705 residue in human MCF7 cells preincubated for 1 hr followed by IL-6 stimulation and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50541369(CHEMBL4635140)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of IL-6 induced STAT3 phosphorylation at Tyr705 residue in human MCF7 cells preincubated for 1 hr followed by IL-6 stimulation and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460520(CHEMBL4228293)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460517(CHEMBL4227185)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50541367(CHEBI:66028 | CHEMBL392591)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of IL-6 induced STAT3 phosphorylation at Tyr705 residue in human MCF7 cells preincubated for 1 hr followed by IL-6 stimulation and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50541368(CHEMBL611361)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of IL-6 induced STAT3 phosphorylation at Tyr705 residue in human MCF7 cells preincubated for 1 hr followed by IL-6 stimulation and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268191(CHEMBL4102765)
Affinity DataIC50:  2.43E+3nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460524(CHEMBL4225893)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50460522(CHEMBL4226829)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50460517(CHEMBL4227185)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human placenta topoisomerase 2alpha assessed as reduction in pBR322 supercoiled DNA relaxation after 30 mins by ethidium bromide staini...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268183(CHEMBL4080410)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kindai University

Curated by ChEMBL
LigandPNGBDBM50268183(CHEMBL4080410)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse HDAC6 expressed in HEK293T cells co-expressing mouse HDA2 using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50268183(CHEMBL4080410)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human HDAC1 expressed in HEK293T cells using Ac-KGLGK(Ac)-MCA as substrate after 30 mins in presence of DTT by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50483440(Moverastin A)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268184(CHEMBL4060026)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268183(CHEMBL4080410)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of human placenta topoisomerase 2alpha assessed as reduction in pBR322 supercoiled DNA relaxation after 30 mins by ethidium bromide staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50460525(CHEMBL4228731)
Affinity DataIC50:  2.61E+4nMAssay Description:Inhibition of human placenta topoisomerase 2alpha assessed as reduction in pBR322 supercoiled DNA relaxation after 30 mins by ethidium bromide staini...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268190(CHEMBL4099888)
Affinity DataIC50:  3.52E+4nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50127140((-)-etoposide | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-d...)
Affinity DataIC50:  5.02E+4nMAssay Description:Inhibition of human placenta topoisomerase 2alpha assessed as reduction in pBR322 supercoiled DNA relaxation after 30 mins by ethidium bromide staini...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50460519(CHEMBL4226061)
Affinity DataIC50:  5.53E+4nMAssay Description:Inhibition of human placenta topoisomerase 2alpha assessed as reduction in pBR322 supercoiled DNA relaxation after 30 mins by ethidium bromide staini...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268187(CHEMBL4104323)
Affinity DataIC50:  5.57E+4nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50127140((-)-etoposide | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-d...)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50268185(CHEMBL4088260)
Affinity DataIC50:  6.45E+4nMAssay Description:Inhibition of recombinant human DNA topoisomerase-2alpha assessed as decrease in relaxation of supercoiled pBR322 DNA after 30 mins by ethidium bromi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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