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Found 87 Enz. Inhib. hit(s) with Target = 'NF-kappa-B inhibitor alpha'
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437341(WITHANOLIDE E)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437352(CHEMBL2408033)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50378033(PHYSALIN F)
Affinity DataIC50:  2.71E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437349(25-HYDROXY PHYSALIN F)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50378034(CHEMBL504404 | NSC-287088 | PHYSALIN B)
Affinity DataIC50:  3.75E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437346(CHEMBL2408037)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437347(PHYSALIN J)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437348(25-HYDROXY PHYSALIN J)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437350(CHEMBL2408034)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437351(PHYSALIN A)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437345(PHYSALIN O)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437344(WITHANOLIDE F)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437343(CHEMBL2333678)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437342(CHEMBL2333675)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437339(CHEMBL2408039)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437340(CHEMBL2408038)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372493(CHEMBL404128)
Affinity DataEC50:  1.30E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataEC50:  1.00E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataEC50:  5.20E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells assessed as ratio of green light emiting IkappaBalpha-fused luciferase expression to r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372494(CHEMBL273148)
Affinity DataEC50:  8.90E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372495(CHEMBL273147)
Affinity DataEC50:  3.70E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372496(CHEMBL273149)
Affinity DataEC50:  1.40E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372497(CHEMBL270798)
Affinity DataEC50:  7.00E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372498(CHEMBL429599)
Affinity DataEC50:  1.10E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372499(CHEMBL270799)
Affinity DataEC50:  4.10E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372500(CHEMBL272553)
Affinity DataEC50:  1.30E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372501(CHEMBL271669)
Affinity DataEC50:  500nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  2.20E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372502(CHEMBL256403)
Affinity DataEC50:  1.40E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372503(CHEMBL401504)
Affinity DataEC50:  5.90E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372504(CHEMBL257446)
Affinity DataEC50:  2.70E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372505(CHEMBL401505)
Affinity DataEC50:  9.40E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372506(CHEMBL256061)
Affinity DataEC50:  4.00E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372507(CHEMBL256062)
Affinity DataEC50:  1.10E+4nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372508(CHEMBL256244)
Affinity DataEC50:  2.00E+4nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372509(CHEMBL256243)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372510(CHEMBL269942)
Affinity DataEC50:  6.80E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372511(CHEMBL404588)
Affinity DataEC50:  3.60E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372512(CHEMBL429586)
Affinity DataEC50:  1.00E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM53740(2-[(5-chloro-4-tosyl-thiazol-2-yl)amino]ethyl-dime...)
Affinity DataEC50:  6.80E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372513(CHEMBL256204)
Affinity DataEC50:  6.80E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM60287(2-nitro-N-(8-quinolinyl)benzenesulfonamide | 2-nit...)
Affinity DataEC50:  1.10E+4nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372514(CHEMBL540966)
Affinity DataEC50:  6.50E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372494(CHEMBL273148)
Affinity DataEC50:  7.20E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells assessed as ratio of green light emiting IkappaBalpha-fused luciferase expression to r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372515(CHEMBL403333)
Affinity DataEC50:  8.00E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372516(CHEMBL272552)
Affinity DataEC50:  700nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372517(CHEMBL256609)
Affinity DataEC50:  6.10E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372518(CHEMBL257234)
Affinity DataEC50:  5.30E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372519(CHEMBL258314)
Affinity DataEC50:  8.00E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50372521(CHEMBL403922)
Affinity DataEC50: >2.00E+4nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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