Compile Data Set for Download or QSAR
maximum 50k data
Found 110 of ic50 for UniProtKB: A0A024R8E4
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560065(CHEMBL4777235)
Affinity DataIC50:  0nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560066(CHEMBL4787034)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50542790(CHEMBL4647584)
Affinity DataIC50:  82nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50542793(CHEMBL4635903)
Affinity DataIC50:  84nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560066(CHEMBL4787034)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553050(CHEMBL4744916)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560066(CHEMBL4787034)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553068(CHEMBL4761806)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50542789(CHEMBL4647726)
Affinity DataIC50:  130nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50:  158nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50542792(CHEMBL4636288)
Affinity DataIC50:  200nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560066(CHEMBL4787034)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560065(CHEMBL4777235)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560065(CHEMBL4777235)
Affinity DataIC50:  230nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50542788(CHEMBL4645959)
Affinity DataIC50:  260nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50593123(GENZ-682452 | GZ-402671 | GZ/SAR402671 | GZ402671 ...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human NTMT1 in human HCT116 cells assessed as reduction in me3-SET level incubated for 72 hrs by western blot analysisMore data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50593123(GENZ-682452 | GZ-402671 | GZ/SAR402671 | GZ402671 ...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human NTMT1 in human HCT116 cells assessed as reduction in me3-RCC1 level incubated for 72 hrs by western blot analysisMore data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50542791(CHEMBL4633108)
Affinity DataIC50:  320nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553069(CHEMBL4796649)
Affinity DataIC50:  340nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553058(CHEMBL4740501)
Affinity DataIC50:  340nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50523491(CHEMBL4475410)
Affinity DataIC50:  414nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM60981((2,3-diphenyl-1,2,4-thiadiazol-5-ylidene)-methyl-a...)
Affinity DataIC50:  460nMAssay Description:Inhibition of full length His-NTMT1 (1 to 222 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as SAH production by Mtase...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553065(CHEMBL4792508)
Affinity DataIC50:  470nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50523490(CHEMBL4575245)
Affinity DataIC50:  485nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553062(CHEMBL4742945)
Affinity DataIC50:  490nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50593123(GENZ-682452 | GZ-402671 | GZ/SAR402671 | GZ402671 ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of full length NTMT1 (1 to 222 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as SAH production by SAHH-coup...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50593123(GENZ-682452 | GZ-402671 | GZ/SAR402671 | GZ402671 ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of full length NTMT1 (1 to 222 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as SAH production by SAHH-coup...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50593123(GENZ-682452 | GZ-402671 | GZ/SAR402671 | GZ402671 ...)
Affinity DataIC50:  560nMAssay Description:Inhibition of full length NTMT1 (1 to 222 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as SAH production by SAHH-coup...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50593123(GENZ-682452 | GZ-402671 | GZ/SAR402671 | GZ402671 ...)
Affinity DataIC50:  560nMAssay Description:Inhibition of full length NTMT1 (1 to 222 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using GPKRIA as substrate preincubated ...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553066(CHEMBL4764028)
Affinity DataIC50:  580nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553064(CHEMBL4756093)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553053(CHEMBL4751006)
Affinity DataIC50:  680nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560065(CHEMBL4777235)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560065(CHEMBL4777235)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553067(CHEMBL4781749)
Affinity DataIC50:  740nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553055(CHEMBL4751138)
Affinity DataIC50:  780nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560066(CHEMBL4787034)
Affinity DataIC50:  800nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50523488(CHEMBL4468450)
Affinity DataIC50:  810nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553061(CHEMBL4745007)
Affinity DataIC50:  840nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553054(CHEMBL4796778)
Affinity DataIC50:  880nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553051(CHEMBL4797618)
Affinity DataIC50:  890nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  890nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50560066(CHEMBL4787034)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50553049(CHEMBL4757419)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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