Found 9 Enz. Inhib. hit(s) with Target = 'N-terminal Xaa-Pro-Lys N-methyltransferase 1' and Ligand = 'BDBM50553049'
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKd: 3.00E+3nMAssay Description:Binding affinity to recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) by ITC assayMore data for this Ligand-Target Pair