Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50014872
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148588(CHEMBL325304 | Heptyl-phosphonic acid monoethyl es...)
Affinity DataIC50:  1.06E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148590((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  1.31E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148587(CHEMBL326268 | Heptyl-phosphonic acid mono-[2-(1,3...)
Affinity DataIC50:  1.47E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148586(Butyl-phosphonic acid ethyl ester 3-phenoxy-benzyl...)
Affinity DataIC50:  2.01E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148593(CHEMBL119521 | Hexyl-phosphonic acid monoethyl est...)
Affinity DataIC50:  3.56E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148585(CHEMBL418868 | Hexyl-phosphonic acid mono-[2-(1,3-...)
Affinity DataIC50:  4.39E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148594((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148583(CHEMBL325149 | Nonyl-phosphonic acid ethyl ester 3...)
Affinity DataIC50:  1.48E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148596(CHEMBL278017 | Heptyl-phosphonic acid ethyl ester ...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148582(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-ethylet...)
Affinity DataIC50:  2.57E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148597((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyleth...)
Affinity DataIC50:  4.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148584(CHEMBL118790 | Hexyl-phosphonic acid ethyl ester 3...)
Affinity DataIC50:  4.26E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148591(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-ethyl e...)
Affinity DataIC50:  5.07E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148592((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  8.71E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148589(Butyl-phosphonic acid monoethyl ester | CHEMBL1182...)
Affinity DataIC50:  4.31E+5nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148595(CHEMBL119480 | Nonyl-phosphonic acid monoethyl est...)
Affinity DataIC50:  4.71E+5nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148581(CHEMBL119236 | Tetradecyl-phosphonic acid ethyl es...)
Affinity DataIC50:  8.62E+5nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed