Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50016594
TargetSphingosine kinase 2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataKi: 9.80E+3nMAssay Description:Binding affinity to recombinant SphK2 (unknown origin) ADP Quest assay systemMore data for this Ligand-Target Pair
TargetAlpha-1-antitrypsin-related protein(Homo sapiens)
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to ATR (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of LCK (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Inhibition of CamK-II (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of MEK 1/2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
Target1-phosphatidylinositol 3-phosphate 5-kinase(Homo sapiens)
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of PIKFYVE (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
Target1-phosphatidylinositol 3-phosphate 5-kinase(Homo sapiens)
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of PIKFYVE (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of MEK 1/2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK6 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Target1-phosphatidylinositol 3-phosphate 5-kinase(Homo sapiens)
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of PIKFYVE (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8/9(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of JNK1/2 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of SAPK2a/p38 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of MEK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK6 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 108nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of Cdk9 (unknown origin) incubated fro 2 hrs by measuring remaining ATP by kinase GloMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TrKA (unknown origin)More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)
Curated by ChEMBL
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of GRK2 (unknown origin)More data for this Ligand-Target Pair
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