Compile Data Set for Download or QSAR
maximum 50k data
Found 386 of ic50 data for polymerid = 1808,50000876
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170371(5-Piperidin-1-ylmethyl-thiazole-4-carboxylic acid ...)
Affinity DataIC50:  75nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267199(CHEMBL4079583)
Affinity DataIC50:  100nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169672(5-(Cyclopentanecarbonyl-amino)-thiazole-4-carboxyl...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129648(3-(4-Methyl-pent-3-enoylamino)-pyridine-2-carboxyl...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170369(5-(2-Ethoxy-3-methyl-butyl)-thiazole-4-carboxylic ...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129642(CHEMBL86427 | Phenyl-acetic acid 2-(thiazol-2-ylca...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169671(5-Propionylamino-thiazole-4-carboxylic acid thiazo...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170363(5-[2-(2-Chloro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50:  230nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169669(5-(Cyclobutanecarbonyl-amino)-thiazole-4-carboxyli...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170383(5-[2-(2-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50:  270nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170370(5-[2-Methoxy-2-(4-methoxy-phenyl)-ethyl]-thiazole-...)
Affinity DataIC50:  310nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129669(3-(5-Methyl-hex-4-enoylamino)-pyridine-2-carboxyli...)
Affinity DataIC50:  310nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129635(3-Formylamino-pyridine-2-carboxylic acid thiazol-2...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129649(CHEMBL315098 | Cyclohexanecarboxylic acid 2-(thiaz...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170358(5-[2-(3-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50:  340nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM17849(3-(2,2-dimethylpropanamido)-N-(1,3-thiazol-2-yl)py...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129672(3-Propionylamino-pyridine-2-carboxylic acid thiazo...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against Saccharomyces cerevisiae methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129672(3-Propionylamino-pyridine-2-carboxylic acid thiazo...)
Affinity DataIC50:  350nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170365(5-Pyrrolidin-1-ylmethyl-thiazole-4-carboxylic acid...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50435227(CHEMBL2392772)
Affinity DataIC50:  360nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM17589((2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxy-N-[(1S...)
Affinity DataIC50:  370nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169656(5-(2-Methyl-but-3-enoylamino)-thiazole-4-carboxyli...)
Affinity DataIC50:  370nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM17589((2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxy-N-[(1S...)
Affinity DataIC50:  370nMAssay Description:Inhibitory activity against human methionine aminopeptidase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129663(3-But-3-enoylamino-pyridine-2-carboxylic acid thia...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129650(CHEMBL314448 | Propionic acid 2-(thiazol-2-ylcarba...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170366(5-[2-(4-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50:  390nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129641(2-Methyl-but-2-enoic acid 2-(thiazol-2-ylcarbamoyl...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM17847(CHEMBL327579 | pyridine-2-carboxylic acid inhibito...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170389(5-(2-Cyclohexyl-2-methoxy-ethyl)-thiazole-4-carbox...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170361(5-(2-Piperidin-1-yl-ethyl)-thiazole-4-carboxylic a...)
Affinity DataIC50:  410nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170382(5-(2-Methoxy-2-phenyl-ethyl)-thiazole-4-carboxylic...)
Affinity DataIC50:  440nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170381(5-(2-Methoxy-hexyl)-thiazole-4-carboxylic acid thi...)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170384(5-((S)-2-Methoxy-2-phenyl-ethyl)-thiazole-4-carbox...)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170388(5-((R)-2-Methoxy-2-phenyl-ethyl)-thiazole-4-carbox...)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169686(5-(4-Fluoro-benzoylamino)-thiazole-4-carboxylic ac...)
Affinity DataIC50:  480nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129646(3-Methyl-but-2-enoic acid 2-(thiazol-2-ylcarbamoyl...)
Affinity DataIC50:  490nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170360(5-(2-Methoxy-4-methyl-pentyl)-thiazole-4-carboxyli...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169679(5-(2-Methoxy-3-methyl-butyl)-thiazole-4-carboxylic...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169679(5-(2-Methoxy-3-methyl-butyl)-thiazole-4-carboxylic...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170374(5-[2-(3-Chloro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50:  520nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129675(2-Methoxy-benzoic acid 2-(thiazol-2-ylcarbamoyl)-p...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170380(Benzyloxy-acetic acid 2-[4-(thiazol-2-ylcarbamoyl)...)
Affinity DataIC50:  550nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170378(5-[2-(4-Chloro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50:  570nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170367(5-[2-Methoxy-2-(2-methoxy-phenyl)-ethyl]-thiazole-...)
Affinity DataIC50:  570nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50435224(CHEMBL2392893)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50435217(CHEMBL2392900)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129656(3-Hexanoylamino-pyridine-2-carboxylic acid thiazol...)
Affinity DataIC50:  620nMAssay Description:Inhibitory concentration against Saccharomyces cerevisiae methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129656(3-Hexanoylamino-pyridine-2-carboxylic acid thiazol...)
Affinity DataIC50:  620nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169670(5-Phenethyl-thiazole-4-carboxylic acid thiazol-2-y...)
Affinity DataIC50:  660nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Shanghai Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50169685(CHEMBL360353 | N-[4-(Thiazol-2-ylcarbamoyl)-thiazo...)
Affinity DataIC50:  670nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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