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Found 10 Enz. Inhib. hit(s) with all data for entry = 1595
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332408(US10196353, Example 52 | US11299457, Example 52)
Affinity DataIC50:  15.8nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332406(US10196353, Example 32 | US11299457, Example 32)
Affinity DataIC50:  31.6nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332402(US10196353, Example 17 | US11299457, Example 17)
Affinity DataIC50:  79.4nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332405(US10196353, Example 27 | US11299457, Example 27)
Affinity DataIC50:  79.4nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332052(US10196353, Example 2 | US11299457, Example 2)
Affinity DataIC50:  100nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332404(US10196353, Example 22 | US11299457, Example 22)
Affinity DataIC50:  158nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332401(US10196353, Example 12 | US11299457, Example 12)
Affinity DataIC50:  251nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332403(US10196353, Example 21 | US11299457, Example 21)
Affinity DataIC50:  316nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332407(US10196353, Example 43 | US11299457, Example 43)
Affinity DataIC50:  631nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM332400(US10196353, Example 7 | US11299457, Example 7)
Affinity DataIC50:  631nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent